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A Selective Inverse Agonist for Central Cannabinoid Receptor Inhibits Mitogen-activated Protein Kinase Activation Stimulated by Insulin or Insulin-like Growth Factor 1

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Constitutively active 5-hydroxytryptamine2C receptors reveal novel inverse agonist activity of receptor ligands.

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Partial agonists, full agonists, antagonists: dilemmas of definition

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Negative antagonists promote an inactive conformation of the beta 2-adrenergic receptor.

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Antagonists of bradykinin that stabilize a G-protein-uncoupled state of the B2 receptor act as inverse agonists in rat myometrial cells

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The Stability of the Agonist β₂-Adrenergic Receptor-G_sComplex: Evidence for Agonist-Specific States

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Identification of a Conserved Switch Residue Responsible for Selective Constitutive Activation of the β2-Adrenergic Receptor

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Brain Purines in a Genetic Mouse Model of Lesch‐Nyhan Disease

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Spontaneous β₂-Adrenergic Signaling Fails To Modulate L-Type Ca²⁺Current in Mouse Ventricular Myocytes

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The C-Terminus of the Prostaglandin-E-Receptor EP3 Subtype is Essential for Activation of GTP-Binding Protein

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Inverse agonistic effect of ICI-174,864 on the cloned delta-opioid receptor: role of G protein and adenylyl cyclase activation.

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Deletion analysis of the m4 muscarinic acetylcholine receptor

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Activation of GTP formation and high-affinity GTP hydrolysis by mastoparan in various cell membranes

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Evidence for nucleoside diphosphokinase-dependent channeling of guanosine 5'-(gamma-thio)triphosphate to guanine nucleotide-binding proteins.

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3H-naloxone benzoylhydrazone binding in MOR-1-transfected Chinese hamster ovary cells: evidence for G-protein-dependent antagonist binding.

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The C Terminal Tail of the Histamine H₂ Receptor Contains Positive and Negative Signals Important for Signal Transduction and Receptor Down‐Regulation

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Is the R and R* dichotomy real?

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Is the R and R∗ dichotomy real?

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