WAY100135: a novel, selective antagonist at presynaptic and postsynaptic 5-HT1A receptors

The rat brain: A stereotaxic atlas of the forebrain and lower parts of the brain stem

1986 • 4,155 citations

Proposals for the classification and nomenclature of functional receptors for 5-hydroxytryptamine

1986 • 1,255 citations

8-Hydroxy-2-(di-n-propylamino)-tetralin discriminates between subtypes of the 5-HT1 recognition site

1983 • 869 citations

The involvement of subtypes of the 5-HT1 receptor and of catecholaminergic systems in the behavioural response to 8-hydroxy-2-(di-n-Propylamino) tetralin in the rat

1984 • 678 citations

Serotonergic component of neuroleptic receptors

1978 • 621 citations

8-hydroxy-2-(di-n-propylamino)tetralin, 8-OH-DPAT, a potent and selective simplified ergot congener with central 5-HT-receptor stimulating activity

1982 • 517 citations

Characterization of alpha 1-adrenergic receptor subtypes in rat brain: a reevaluation of [3H]WB4104 and [3H]prazosin binding.

1986 • 456 citations

A nonclassical 5-hydroxytryptamine receptor positively coupled with adenylate cyclase in the central nervous system.

1988 • 435 citations

The concept of selectivity in 5-HT receptor research

1990 • 425 citations

Lysergic acid diethylamide and serotonin: a comparison of effects on serotonergic neurons and neurons receiving a serotonergic input.

1974 • 311 citations

(-)-Propranolol blocks the inhibition of serotonergic dorsal raphe cell firing by 5-HT1A selective agonists

1986 • 301 citations

Subtypes of Receptors for Serotonin

1990 • 199 citations

Chemical Protection against Ionizing Radiation: I. Sampling Methods for Screening Compounds in Radiation Protection Studies with Mice

1957 • 186 citations

NAN-190: an arylpiperazine analog that antagonizes the stimulus effects of the 5-HT1A agonist 8-hydroxy-2-(di-n-propylamino) tetralin (8-OH-DPAT)

1988 • 183 citations

Direct evidence for an important species difference in the mechanism of 8‐OH‐DPAT‐induced hypothermia

1991 • 174 citations

Centrally acting hypotensive agents with affinity for 5‐HT_1A binding sites inhibit forskolin‐stimulated adenylate cyclase activity in calf hippocampus

1988 • 151 citations

Mixed agonist/antagonist properties of NAN-190 at 5-HT1A Receptors: Behavioural and in vivo brain microdialysis studies

1990 • 133 citations

BMY 7378, a buspirone analog with high affinity, selectivity and low intrinsic activity at the 5-HT1A receptor in rat and guinea pig hippocampal membranes

1987 • 128 citations

Buspirone: Action on serotonin receptors in calf hippocampus

1983 • 127 citations

Further investigation of the in vivo pharmacological properties of the putative 5-HT1A antagonist, BMY 7378

1990 • 109 citations

Intrinsic activity of enantiomers of 8-hydroxy-2-(di-n-propylamino)tetralin and its analogs at 5-hydroxytryptamine1A receptors that are negatively coupled to adenylate cyclase.

1991 • 106 citations

Spiroxatrine: A selective serotonin1A receptor antagonist

1986 • 104 citations

Agonist/antagonist interactions with cloned human 5-HT1A receptors: variations in intrinsic activity studied in transfected HeLa cells

1992 • 104 citations

3H-DOB (4-bromo-2,5-dimethoxyphenylisopropylamine) labels a guanyl nucleotide-sensitive state of cortical 5-HT2 receptors.

1987 • 103 citations

Pharmacology of the novel 5-hydroxytryptamine1A receptor antagonist (S)-5-fluoro-8-hydroxy-2-(dipropylamino)tetralin: inhibition of (R)-8-hydroxy-2-(dipropylamino)tetralin-induced effects.

1991 • 100 citations

Arylpiperazine derivatives as high-affinity 5-HT1A serotonin ligands

1988 • 98 citations

Pharmacological analysis of muscarinic receptors coupled to oxyntic cell secretion in the mouse stomach

1985 • 91 citations

Blockade of the central 5-HT autoreceptor by β-adrenoceptor antagonists

1986 • 90 citations

The putative 5-HT1A receptor antagonists NAN-190 and BMY 7378 are partial agonists in the rat dorsal raphe nucleus in vitro

1992 • 84 citations

Effect of the putative 5-HT1A receptor antagonist NAN-190 on rat brain serotonergic transmission

1991 • 54 citations

Stereoselective blockade of central [3H]5-hydroxytryptamine binding to multiple sites (5-HT1A, 5-HT1B and 5-HT1C) by mianserin and propranolol

1987 • 50 citations

Heterogeneos 3H-rauwolscine binding sites in rat cortex: Two alpha2-adrenoceptor subtypes or an additional non-adrenergic interaction?

1988 • 42 citations

[3H]8-OH-DPAT labels the 5-Hydroxytryptamine uptake recognition site and the 5-HT1A binding site in the rat striatum

1988 • 38 citations

The novel 5-HT1A receptor antagonist (S)-UH-301 prevents (R)-8-OH-DPAT-induced decrease in interstitial concentrations of serotonin in the rat hippocampus

1992 • 36 citations

Distinctions between ligand-binding sites for [3H]dopamine and D2 dopaminergic receptors characterized with [3H]spiroperidol.

1984 • 20 citations