Deletion of the Serotonin 5-HT2C Receptor PDZ Recognition Motif Prevents Receptor Phosphorylation and Delays Resensitization of Receptor Responses

Regulation of serotonin-2C receptor G-protein coupling by RNA editing

1997 • 985 citations

A kinase-regulated PDZ-domain interaction controls endocytic sorting of the β2-adrenergic receptor

1999 • 673 citations

RNA Editing of the Human Serotonin 5-Hydroxytryptamine 2C Receptor Silences Constitutive Activity

1999 • 353 citations

Functional characterization of agonists at recombinant human 5‐HT_2A, 5‐HT_2B and 5‐HT_2C receptors in CHO‐K1 cells

1999 • 347 citations

A unique serotonin receptor in choroid plexus is linked to phosphatidylinositol turnover.

1986 • 265 citations

Constitutively active 5-hydroxytryptamine2C receptors reveal novel inverse agonist activity of receptor ligands.

1994 • 249 citations

Serotonin 5‐HT_2C Receptor RNA Editing Alters Receptor Basal Activity

1999 • 180 citations

Truncation of the receptor carboxyl terminus impairs agonist-dependent phosphorylation and desensitization of the alpha 1B-adrenergic receptor.

1994 • 132 citations

Identification, molecular cloning, and distribution of a short variant of the 5-hydroxytryptamine2C receptor produced by alternative splicing.

1996 • 130 citations

Characterization of the Phosphorylation Sites Involved in G Protein-coupled Receptor Kinase- and Protein Kinase C-mediated Desensitization of the α1B-Adrenergic Receptor

1997 • 123 citations

Ligand-induced Desensitization of the Human CXC Chemokine Receptor-2 Is Modulated by Multiple Serine Residues in the Carboxyl-terminal Domain of the Receptor

1997 • 119 citations

The Human Serotonin 5-HT2CReceptor: Complete cDNA, Genomic Structure, and Alternatively Spliced Variant

1996 • 107 citations

Dissecting G Protein-coupled Receptor Signaling Pathways with Membrane-permeable Blocking Peptides

2000 • 88 citations

Role of cytoplasmic tail phosphorylation sites of platelet-activating factor receptor in agonist-induced desensitization.

1994 • 80 citations

C-terminal Truncation of the Neurokinin-2 Receptor Causes Enhanced and Sustained Agonist-induced Signaling

1995 • 76 citations

Desensitization of N-Formylpeptide Receptor-mediated Activation Is Dependent upon Receptor Phosphorylation

1997 • 70 citations

Agonist-Induced Phosphorylation of the Angiotensin AT_1aReceptor Is Localized to a Serine/Threonine-Rich Region of Its Cytoplasmic Tail

1998 • 70 citations

Increased basal phosphorylation of the constitutively active serotonin 2C receptor accompanies agonist-mediated desensitization.

1995 • 70 citations

Roles of Cholecystokinin Receptor Phosphorylation in Agonist-Stimulated Desensitization of Pancreatic Acinar Cells and Receptor-Bearing Chinese Hamster Ovary Cholecystokinin Receptor Cells

1997 • 40 citations

Identification of rat serotonin 5-HT2C receptors as glycoproteins containing N-linked oligosaccharides

1995 • 36 citations

Role of C-terminal Serines in Desensitization and Phosphorylation of the Mouse Thromboxane Receptor

1998 • 35 citations

Generation of anti-peptide antibodies against serotonin 5-HT2A and 5-HT2C receptors

1997 • 30 citations

Serotonin elevates intracellular Ca2+ in rat choroid plexus epithelial cells by acting on 5-HT2C receptors

1995 • 28 citations

Rapid Desensitization of Serotonin 5‐HT_2C Receptor‐Stimulated Intracellular Calcium Mobilization in CHO Cells Transfected with Cloned Human 5‐HT_2C Receptors

1995 • 28 citations

Characterization of N- and C-terminal deletion mutants of the rat serotonin HT2 receptor in Xenopus laevis oocytes

1991 • 26 citations

Comparative desensitization of the human 5‐HT_2A and 5‐HT_2C receptors expressed in the human neuroblastoma cell line SH‐SY5Y

1998 • 26 citations

Calcineurin inhibits desensitization of cloned rat 5-HT1C receptors

1993 • 19 citations