[3H]‐MK 912 binding delineates two α2‐adrenoceptor subtypes in rat CNS one of which is identical with the cloned pA2d α2‐adrenoceptor
Data up to Jan 2025
Total Citations Per Year
Abstract
References (38)
PROTEIN MEASUREMENT WITH THE FOLIN PHENOL REAGENT
1951 • 319,299 citations
A STUDY OF THE ADRENOTROPIC RECEPTORS
1948 • 2,856 citations
A functional basis for classification of α-adrenergic receptors
1977 • 802 citations
Cloning, Sequencing, and Expression of the Gene Coding for the Human Platelet α 2 -Adrenergic Receptor
1987 • 792 citations
Differentiation of receptors responsive to isoproterenol
1967 • 484 citations
Cloning and expression of a human kidney cDNA for an alpha 2-adrenergic receptor subtype.
1988 • 440 citations
Alpha-2A and alpha-2B adrenergic receptor subtypes: antagonist binding in tissues and cell lines containing only one subtype.
1988 • 307 citations
Heterogeneity of alpha-2 adrenergic receptors
1985 • 297 citations
Expansion of the alpha 2-adrenergic receptor family: cloning and characterization of a human alpha 2-adrenergic receptor subtype, the gene for which is located on chromosome 2.
1990 • 287 citations
An aspartate conserved among G-protein receptors confers allosteric regulation of alpha 2-adrenergic receptors by sodium.
1990 • 266 citations
Isolation of rat genomic clones encoding subtypes of the alpha 2-adrenergic receptor. Identification of a unique receptor subtype
1991 • 220 citations
Pharmacological classification of adrenergic α receptors in the guinea pig
1978 • 164 citations
Molecular characterization of a rat alpha 2B-adrenergic receptor.
1990 • 163 citations
Molecular characterization of α1- and α2-adrenoceptors
1991 • 153 citations
Delineation of rat kidney α2A- and α2B-adrenoeeptors with [3H]RX821002 radiollgand binding: computer modelling reveals that guanfacine is an α2A-selective compound
1991 • 137 citations
Expression of three alpha 2-adrenergic receptor subtypes in rat tissues: implications for alpha 2 receptor classification.
1990 • 131 citations
Agonist versus antagonist binding to alpha-adrenergic receptors.
1980 • 118 citations
Characterization of the alpha-2C adrenergic receptor subtype in the opossum kidney and in the OK cell line.
1991 • 116 citations
Characterization of alpha-2 adrenergic receptors in the OK cell, an opossum kidney cell line.
1988 • 112 citations
Pharmacological characterization of rat alpha 2-adrenergic receptors.
1991 • 110 citations
Distribution of α2-adrenergic receptor mRNAs in the rat CNS
1991 • 109 citations
Novel α2-adrenoceptor antagonists show selectivity for α2A- and α2B-adrenoceptor subtypes
1989 • 109 citations
Further Characterization of the Guinea Pig Cerebral Cortex Idazoxan Receptor: Solubilization, Distinction from the Imidazole Site, and Demonstration of Cirazoline as an Idazoxan Receptor‐Selective Drug
1990 • 103 citations
Interactions of Agonists with Platelet α2-Adrenergic Receptors
1982 • 102 citations
Rat Spinal Cord α2‐Adrenoceptors are of the α2A‐Subtype: Comparison with α2A‐ and α2B‐Adrenoceptors in Rat Spleen, Cerebral Cortex and Kidney Using 3H‐RX821002 Ligand Binding
1991 • 79 citations
Molecular cloning, sequencing and expression of an ?2-adrenergic receptor complementary DNA from rat brain
1990 • 68 citations
Delineation of three pharmacological subtypes of α2‐adrenoceptor in the rat kidney
1991 • 60 citations
α2-Adrenoceptors in rat hypothalamus and cerebral cortex: functional evidence for pharmacologically distinct subpopulations
1985 • 58 citations
The rat α2‐C4 adrenergic receptor gene encodes a novel pharmacological subtype
1991 • 51 citations
Heterogeneos 3H-rauwolscine binding sites in rat cortex: Two alpha2-adrenoceptor subtypes or an additional non-adrenergic interaction?
1988 • 42 citations
Adrenoceptors: Structure, Mechanisms, Function
1991 • 39 citations
Heterogeneity of α2‐adrenoceptors in rat cortex but not human platelets can be defined by 8‐OH‐DPAT, RU 24969 and methysergide
1990 • 33 citations
[3H]L-657, 743 (MK-912): A new, high affinity, selective radioligand for brain α2-adrenoceptors
1989 • 29 citations
Agonist binding at alpha2-adrenoceptors of human platelets using 3H-UK-14,304: regulation by Gpp(NH)p and cations
1987 • 26 citations
Antinociceptive Actions of α2‐Adrenoceptor Agonists in the Rat Spinal Cord: Evidence for Antinociceptive α2‐Adrenoceptor Subtypes and Dissociation of Antinociceptive α2‐Adrenoceptors from Cyclic AMP
1990 • 23 citations
Differential blockade by (?)mianserin of the alpha2-adrenoceptors mediating inhibition of noradrenaline and serotonin release from rat brain synaptosomes
1983 • 19 citations
Pharmacological evidence for alpha 2c and alpha 2d adrenergic receptor subtypes
1991 • 12 citations
Structural and Pharmacological Differences between Codfish and Rat Brain α1‐Adrenergic Receptors Revealed by Photoaffinity Labeling with 125I‐APDQ
1986 • 9 citations