cis-2,4-methanoglutamate is a potent and selective N-methyl-D-aspartate receptor agonist

Simultaneous analysis of families of sigmoidal curves: application to bioassay, radioligand assay, and physiological dose-response curves.

1978 • 2,400 citations

CPP, a new potent and selective NMDA antagonist. Depression of central neuron responses, affinity for [3H]d-AP5 binding sites on brain membranes and anticonvulsant activity

1986 • 311 citations

Excitatory amino acids in health and disease.

1988 • 254 citations

Action of 3-((±)-2-car☐ypiperazin-4-yl)-propyl-1-phosphonic aci (CPP): a new and highly potent antagonist of N-methyl-d-aspartate receptors in the hippocampus

1986 • 239 citations

CPP, a selective N-methyl-D-aspartate (NMDA)-type receptor antagonist: characterization in vitro and in vivo.

1987 • 231 citations

CGS 19755, a selective and competitive N-methyl-D-aspartate-type excitatory amino acid receptor antagonist.

1988 • 219 citations

CNS receptors: From molecular pharmacology to behavior

1983 • 218 citations

Cellular uptake disguises action of L‐glutamate on N‐methyl‐D‐aspartate receptors: With an appendix: Diffusion of transported amino acids into brain slices

1985 • 171 citations

Structure/activity relations of N-methyl-d-aspartate receptor ligands as studied by their inhibition of [3H]d2-amino-5-phosphonopentanoic acid binding in rat brain membranes

1988 • 163 citations

Identification and Characterization of an N‐Methyl‐D‐Aspartate‐Specific L‐[³H]Glutamate Recognition Site in Synaptic Plasma Membranes

1987 • 131 citations

Characterization of Two [³H]Glutamate Binding Sites in Rat Hippocampal Membranes

1981 • 128 citations

Characterization df a [³H]Glycine Recognition Site as a Modulatory Site of the N‐Methyl‐D‐Aspartate Receptor Complex

1989 • 106 citations

Excitatory Amino Acid Receptor Potency and Subclass Specificity of Sulfur-Containing Amino Acids

1987 • 103 citations

Response of Schaffer collateral-CA1 pyramidal cell synapses of the hippocampus to analogues of acidic amino acids

1982 • 98 citations

2,4-Methanoproline (2-carboxy-2,4-methanopyrrolidine) and 2,4-methanoglutamic acid (1-amino-1,3-dicarboxycyclobutane) in seeds of Ateleia herbert smithii Pittier (Leguminosae)

1980 • 90 citations

Classification and properties of acidic amino acid receptors in hippocampus. I. Electrophysiological studies of an apparent desensitization and interactions with drugs which block transmission

1983 • 85 citations

Effects of guanine nucleotides on N-methyl-D-aspartate receptor-ligand interactions.

1988 • 61 citations

1-Aminocyclobutane-1-carboxylate (ACBC): a specific antagonist of the N-methyl-D-aspartate receptor coupled glycine receptor

1989 • 61 citations

Molecular target size analyses of the NMDA-receptor complex in rat cortex

1989 • 51 citations

Pharmacology of the excitatory actions of sulphonic and sulphinic amino acids.

1983 • 48 citations

Regiospecific additions of hydrazoic acid and benzylamine to 1-(arylsulfonyl)bicyclo[1.1.0]Butanes. Application to the synthesis of cis and trans 2,7-methanoglutamic acids

1988 • 34 citations

Glycine antagonist action of 1-aminocyclobutane-1-carboxylate (ACBC) in Xenopus oocytes injected with rat brain mRNA

1989 • 30 citations

Excitation of rat hippocampal neurones by the stereoisomers of cis- and trans-1-amino-1,3-cyclopentane dicarboxylate

1987 • 14 citations