LIMITATIONS OF THE BENZODIAZEPINE RECEPTOR NOMENCLATURE: A PROPOSAL FOR A PHARMACOLOGICAL CLASSIFICATION AS OMEGA RECEPTOR SUBTYPES

Benzodiazepine Receptor: Demonstration in the Central Nervous System

1977 • 1,705 citations

Benzodiazepine receptors in rat brain

1977 • 1,459 citations

The peripheral-type benzodiazepine receptor. Localization to the mitochondrial outer membrane.

1986 • 682 citations

Isolation, characterization, and purification to homogeneity of an endogenous polypeptide with agonistic action on benzodiazepine receptors.

1983 • 631 citations

Urinary and brain beta-carboline-3-carboxylates as potent inhibitors of brain benzodiazepine receptors.

1980 • 542 citations

Quantitative receptor autoradiography using [3H]Ultrofilm: application to multiple benzodiazepine receptors

1982 • 529 citations

Some properties of brain specific benzodiazepine receptors: New evidence for multiple receptors

1979 • 412 citations

Agonist and antagonist benzodiazepine receptor interaction in vitro

1981 • 383 citations

Peripheral benzodiazepine binding sites: Effect of PK 11195, 1-(2-chlorophenyl)-n-methyl-n-(1-methylpropyl)-3-isoquinolinecarboxamide

1983 • 342 citations

Anxiolytic activity of an endogenous adrenal steroid

1986 • 317 citations

Porphyrins are endogenous ligands for the mitochondrial (peripheral-type) benzodiazepine receptor.

1987 • 297 citations

Specific high-affinity binding sites for [3H]Ro 5-4864 in rat brain and kidney.

1983 • 296 citations

A synthetic non-benzodiazepine ligand for benzodiazepine receptors: A probe for investigating neuronal substrates of anxiety

1979 • 284 citations

Zolpidem, a novel nonbenzodiazepine hypnotic. I. Neuropharmacological and behavioral effects.

1986 • 274 citations

Peripheral-Type Benzodiazepine Receptors in Endocrine Organs: Autoradiographic Localization in Rat Pituitary, Adrenal, and Testis*

1985 • 268 citations

Benzodiazepine Receptor-Mediated Chemotaxis of Human Monocytes

1985 • 239 citations

Peripheral benzodiazepine binding sites: Effect of PK 11195, 1-(2-chlorophenyl)-n-methyl-(1-methylpropyl)-3 isoquinolinecarboxamide

1983 • 230 citations

2-Arylpyrazolo[4,3-c]quinolin-3-ones: a novel agonist, a partial agonist and an antagonist of benzodiazepines

1982 • 215 citations

Ethyl β-carboline-3-carboxylate shows differential benzodiazepine receptor interaction

1980 • 210 citations

Benzodiazepines that bind at peripheral sites inhibit cell proliferation.

1984 • 210 citations

Pharmacological profile of the imidazopyridine zolpidem at benzodiazepine receptors and electrocorticogram in rats

1985 • 168 citations

Ligands for benzodiazepine receptors with positive and negative efficacy

1984 • 157 citations

Interaction of benzodiazepines with mouse macrophages

1984 • 146 citations

Imaging of a glioma using peripheral benzodiazepine receptor ligands.

1987 • 136 citations

Subcellular Localization of “Peripheral‐Type” Binding Sites for Benzodiazepines in Rat Brain

1986 • 135 citations

Autoradiographic Localization of [³H]Zolpidem Binding Sites in the Rat CNS: Comparison with the Distribution of [³H]Flunitrazepam Binding Sites

1987 • 121 citations

Tranquillizers can block mitogenesis in 3T3 cells and induce differentiation in Friend cells

1980 • 119 citations

Hypnotic activity of an imidazo‐pyridine (zolpidem).

1986 • 117 citations

Complete amino acid sequences of bovine and human endozepines. Homology with rat diazepam binding inhibitor.

1986 • 114 citations

High affinity [3H]zolpidem binding in the rat brain: an imidazopyridine with agonist properties at central benzodiazepine receptors

1986 • 110 citations

Benzodiazepines have high-affinity binding sites and induce melanogenesis in B16/C3 melanoma cells.

1981 • 95 citations

Affinity of various ligands for benzodiazepine receptors in rat cerebellum and hippocampus

1984 • 92 citations

Demonstration of benzodiazepine-like molecules in the mammalian brain with a monoclonal antibody to benzodiazepines.

1985 • 88 citations

Structural requirements for the binding of benzodiazepines to their peripheral-type sites.

1984 • 73 citations

Benzodiazepine receptors resolved

1986 • 72 citations

Isolation and identification in bovine cerebral cortex of n-butyl beta-carboline-3-carboxylate, a potent benzodiazepine binding inhibitor.

1986 • 71 citations

In vitro characterization of benzodiazepine receptor agonists, antagonists, inverse agonists and agonist/antagonists.

1984 • 68 citations

Distribution of endogenous benzodiazepine receptor ligand-monoamine oxidase inhibitory activity (tribulin) in tissues

1986 • 48 citations

Endogenous benzodiazepine receptor agonist in human and mammalian plasma

1986 • 38 citations

Pharmacokinetic and Dynamic Studies with a New Anxiolytic Imidazo-Pyridine Alpidem Utilizing Pharmaco-EEG and Psychometry

1986 • 36 citations

Characterization of benzodiazepine receptors in the bovine pineal gland: evidence for the presence of an atypical binding site

1986 • 33 citations

ChemInform Abstract: 2‐ARYLPYRAZOLO(4,3‐C)QUINOLIN‐3‐ONES: A NOVEL AGONIST, A PARTIAL AGONIST AND AN ANTAGONIST OF BENZODIAZEPINES

1982 • 29 citations

Benzodiazepine receptors in the human cerebellar cortex: a quantitative autoradiographic and pharmacological study demonstrating the predominance of type I receptors

1987 • 25 citations

High density of [3H]Ro 5-4864 ‘peripheral’ benzodiazepine binding sites in the pineal gland

1984 • 24 citations

PK 11195, an antagonist of peripheral type benzodiazepine receptors, modulates BAY K8644 sensitive but not β- or H2-receptor sensitive voltage operated calcium channels in the guinea pig heart

1986 • 21 citations

Ontogenetic properties of benzodiazepine receptor subtypes in rat spinal cord

1985 • 18 citations

Benzodiazepine receptor sites in bovine pineal

1982 • 9 citations