Ligands for benzodiazepine receptors with positive and negative efficacy

Benzodiazepine receptors in rat brain

1977 • 1,459 citations

Specific benzodiazepine receptors in rat brain characterized by high-affinity (3H)diazepam binding.

1977 • 1,246 citations

Interaction of Convulsive Ligands with Benzodiazepine Receptors

1982 • 549 citations

Urinary and brain beta-carboline-3-carboxylates as potent inhibitors of brain benzodiazepine receptors.

1980 • 542 citations

Some properties of brain specific benzodiazepine receptors: New evidence for multiple receptors

1979 • 412 citations

Molecular heterogeneity of benzodiazepine receptors

1980 • 329 citations

Properties of 3H-diazepam binding to benzodiazepine receptors in rat cerebral cortex

1977 • 323 citations

Specific high-affinity binding sites for [3H]Ro 5-4864 in rat brain and kidney.

1983 • 296 citations

[³H]Propyl ?-Carboline-3-Carboxylate as a Selective Radioligand for the BZ₁Benzodiazepine Receptor Subclass

1981 • 255 citations

Benzodiazepine receptor ligands with positive and negative efficacy

1983 • 244 citations

Ethyl β-carboline carboxylate lowers seizure threshold and antagonizes flurazepam-induced sedation in rats

1981 • 225 citations

2-Arylpyrazolo[4,3-c]quinolin-3-ones: a novel agonist, a partial agonist and an antagonist of benzodiazepines

1982 • 215 citations

β-Carboline-3-carboxylic acid ethyl ester antagonizes diazepam activity

1980 • 193 citations

Anxiogenic and non-anxiogenic benzodiazepine antagonists

1983 • 165 citations

Audiogenic seizures in DBA/2 mice discriminate sensitively between low efficacy benzodazepine receptor agonists and inverse agonists

1983 • 147 citations

GABA reduces binding of 3H-methyl β-carboline-3-carboxylate to brain benzodiazepine receptors

1981 • 126 citations

Does the reversal of the anticonflict effect of phenobarbital by β-CCE and FG 7142 indicate benzodiazepine receptor-mediated anxiogenic properties?

1982 • 105 citations

ANXIETY

1982 • 84 citations

Differential modulation of [35S]TBPS binding by the occupancy of benzodiazepine receptors with its ligands

1983 • 61 citations

Distinction of benzodiazepine agonists from antagonists by photoaffinity labelling of benzodiazepine receptors in vitro

1982 • 54 citations

Anticonvulsant action in the photosensitive baboon, Papio papio, of a novel β-carboline derivative, ZK 91296

1983 • 43 citations