Pharmacological effects of AMPA receptor potentiators LY392098 and LY404187 on rat neuronal AMPA receptors in vitro
Data up to Jan 2025
Total Citations Per Year
Abstract
References (30)
Improved patch-clamp techniques for high-resolution current recording from cells and cell-free membrane patches
1981 • 18,584 citations
Cloned Glutamate Receptors
1994 • 3,989 citations
A Family of AMPA-Selective Glutamate Receptors
1990 • 1,453 citations
The TINS/TiPS Lecture the molecular biology of mammalian glutamate receptor channels
1993 • 882 citations
AMPA receptor subunits expressed by single purkinje cells
1992 • 524 citations
Hippocampal neurons exhibit cyclothiazide-sensitive rapidly desensitizing responses to kainate
1993 • 369 citations
Neuropharmacology of AMPA and kainate receptors
1998 • 362 citations
Calcium buffering properties of calbindin D28k and parvalbumin in rat sensory neurones.
1993 • 348 citations
Kainate receptors are involved in synaptic plasticity
1999 • 328 citations
The differential expression patterns of messenger RNAs encoding non-N-methyl-d-aspartate glutamate receptor subunits (GluR1–4) in the rat brain
1993 • 304 citations
Allosteric potentiation of quisqualate receptors by a nootropic drug aniracetam.
1990 • 303 citations
Cyclothiazide differentially modulates desensitization of alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor splice variants.
1994 • 295 citations
RNA editing of brain glutamate receptor channels: mechanism and physiology1Published on the World Wide Web on 5 February 1998.1
1998 • 263 citations
Modulation of excitatory synaptic transmission by drugs that reduce desensitization at AMPA/kainate receptors
1991 • 252 citations
Diazoxide blocks glutamate desensitization and prolongs excitatory postsynaptic currents in rat hippocampal neurons.
1992 • 123 citations
A centrally active drug that modulates AMPA receptor gated currents
1994 • 111 citations
A Novel Allosteric Potentiator of AMPA Receptors: 4-[2-(Phenylsulfonylamino)ethylthio]-2,6-Difluoro-Phenoxyacetamide
1997 • 104 citations
Pharmacological discrimination of GluR5 and GluR6 kainate receptor subtypes by (3S,4aR,6R,8aR)-6-[2-(1(2)H-tetrazole-5-yl)ethyl]decahyd roisdoquinoline-3 carboxylic-acid.
1996 • 98 citations
2,3‐Benzodiazepines (GYKI 52466 and Analogs): Negative Allosteric Modulators of AMPA Receptors
1996 • 95 citations
Nootropic Drugs Positively Modulate α‐Amino‐3‐Hydroxy‐5‐Methyl‐4‐Isoxazolepropionic Acid‐Sensitive Glutamate Receptors in Neuronal Cultures
1992 • 94 citations
Novel AMPA receptor potentiators LY392098 and LY404187: effects on recombinant human AMPA receptors in vitro
2001 • 79 citations
Biarylpropylsulfonamides as Novel, Potent Potentiators of 2-Amino-3- (5-methyl-3-hydroxyisoxazol-4-yl)- propanoic Acid (AMPA) Receptors
2000 • 73 citations
AMPA receptor heterogeneity in rat hippocampal neurons revealed by differential sensitivity to cyclothiazide
1996 • 71 citations
Adrenaline and extracellular ATP switch between two modes of acid extrusion in the guinea‐pig ventricular myocyte.
1992 • 53 citations
Aniracetam has proportionately smaller effects on synapses expressing long-term potentiation: Evidence that receptor changes subserve LTP
1990 • 50 citations
7-Chloro-3-methyl-3,4-dihydro-2H-1,2,4-benzothiadiazine S,S-dioxide (IDRA 21), a congener of aniracetam, potently abates pharmacologically induced cognitive impairments in patas monkeys.
1995 • 49 citations
Pharmacological characterization of a GluR6 kainate receptor in cultured hippocampal neurons
1999 • 42 citations
LY392098, a novel AMPA receptor potentiator: electrophysiological studies in prefrontal cortical neurons
2001 • 25 citations
The regulation of AMPA receptor-binding sites
1998 • 18 citations
Differential modulation of the GYKI 53784-induced inhibition of AMPA currents by various AMPA-positive modulators in cerebellar Purkinje cells
2000 • 10 citations