5-HT_1D Receptor Agonist Properties of Novel 2-[5-[[(Trifluoromethyl)sulfonyl]oxy]indolyl]ethylamines and Their Use as Synthetic Intermediates

The rat brain in stereotaxic coordinates

1983 • 28,962 citations

LIGAND: A versatile computerized approach for characterization of ligand-binding systems

1980 • 8,534 citations

Axonal regeneration in the rat spinal cord produced by an antibody against myelin-associated neurite growth inhibitors

1990 • 1,232 citations

A practical computer-based approach to the analysis of radioligand binding experiments

1983 • 834 citations

The genomic clone G-21 which resembles a β-adrenergic receptor sequence encodes the 5-HT1A receptor

1988 • 594 citations

Characterization of a novel 3H-5-hydroxytryptamine binding site subtype in bovine brain membranes

1987 • 406 citations

Positive feedback of glutamate exocytosis by metabotropic presynaptic receptor stimulation

1992 • 354 citations

Species differences in the pharmacology of terminal 5-HT autoreceptors in mammalian brain

1989 • 354 citations

Human serotonin 1D receptor is encoded by a subfamily of two distinct genes: 5-HT1D alpha and 5-HT1D beta.

1992 • 293 citations

A single amino-acid difference confers major pharmacological variation between human and rodent 5-HT1B receptors

1992 • 279 citations

CYCLOPENTADIENYL COMPOUNDS OF Sc, Y, La, Ce AND SOME LANTHANIDE ELEMENTS

1954 • 257 citations

A subfamily of 5-HT1D receptor genes

1992 • 230 citations

Molecular pharmacology of 5-HT1D recognition sites: Radioligand binding studies in human, pig and calf brain membranes

1988 • 177 citations

Sumatriptan (GR 43175) interacts selectively with 5-HT1B and 5-HT1D binding sites

1989 • 160 citations

Pustative anxiolytics 8-OH-DPAT, buspirone and TVX Q 7821 are agonists at 5-HT1A autoreceptors in the raphé nuclei

1986 • 128 citations

Clinical and experimental effects of sumatriptan in humans

1993 • 119 citations

substituted (S)-Phenylpiperidines and Rigid Congeners as Preferential Dopamine Autoreceptor Antagonists: Synthesis and Structure-Activity Relationships

1994 • 110 citations

Membrane potential has no direct role in evoking neurotransmitter release

1988 • 102 citations

Evolution of a Novel Series of [(N,N-Dimethylamino)propyl]- and Piperazinylbenzanilides as the First Selective 5-HT1D Antagonists

1994 • 99 citations

Synthesis and Serotonergic Activity of N,N-Dimethyl-2-[5-(1,2,4-triazol-1-ylmethyl)-1H-indol-3-yl]ethylamine and Analogs: Potent Agonists for 5-HT1D Receptors

1995 • 73 citations

Release‐Regulating Serotonin 5‐HT_1D Autoreceptors in Human Cerebral Cortex

1993 • 64 citations

Synthesis and Biological Activity of 3-[2-(Dimethylamino)ethyl]-5-[(1,1-dioxo-5-methyl-1,2,5-thiadiazolidin-2-yl)methyl]-1H-indole and Analogs: Agonists for the 5-HT1D Receptor

1994 • 61 citations

5-HT1 receptors mediating contraction in bovine cerebral arteries: a model for human cerebrovascular ‘5-HT1Dβ‘ receptors

1993 • 59 citations

Stimulation of central 5-HT1D receptors causes hypothermia in the guinea-pig

1994 • 53 citations

Simultaneous measurement of 5-hydroxytryptophan and l-dihydroxyphenylalanine by high-performance liquid chromatography with electrochemical detection

1982 • 51 citations

The activity of 5-HT1D receptor ligands at cloned human 5-HT1Dα and 5-HT1Dβ receptors

1995 • 48 citations

5-[(3-Nitropyrid-2-yl)amino]indoles: Novel Serotonin Agonists with Selectivity for the 5-HT1D Receptor. Variation of the C3 Substituent on the Indole Template Leads to Increased 5-HT1D Receptor Selectivity

1994 • 36 citations

Synthesis and serotonergic activity of arylpiperazide derivatives of serotonin: potent agonists for 5-HT1D receptors

1995 • 35 citations

Indole N-alkylation of tryptamines via dianion and phthalimido intermediates. New potential indolealkylamine haptens

1978 • 28 citations

Azetidinone antibiotics. XV. Synthesis of 2,3-methylenecepham derivatives via intramolecular cyclization of diazosulfoxides

1975 • 25 citations

5‐HT_1D serotonin receptors: Results of a structure‐affinity investigation

1991 • 24 citations

Synthesis and Evaluation of Pharmacological and Pharmacokinetic Properties of Monopropyl Analogs of 5-, 7-, and 8-[[(Trifluoromethyl)sulfonyl]oxy]-2-aminotetralins: Central Dopamine and Serotonin Receptor Activity

1995 • 22 citations

Role of Adenylate Cyclase in the Modulation of the Release of Dopamine: A Microdialysis Study in the Striatum of the Rat

1990 • 22 citations

Galanin: profile of a new neuropeptide

1986 • 13 citations

Atlas of protein side-chain interactions, volumes I and II

1993 • 8 citations

Section Review—Central & Peripheral Nervous Systems: The Evolution of Selective 5-HT_IDReceptor Antagonists

1995 • 3 citations