Determination of the receptor selectivity of opioid agonists in the guinea‐pig ileum and mouse vas deferens by use of β‐funaltrexamine

SOME QUANTITATIVE USES OF DRUG ANTAGONISTS

1959 • 3,948 citations

The effects of morphine- and nalorphine- like drugs in the nondependent and morphine-dependent chronic spinal dog.

1976 • 2,883 citations

Endogenous opioid peptides: multiple agonists and receptors

1977 • 2,494 citations

U-50,488: a selective and structurally novel non-Mu (kappa) opioid agonist.

1983 • 795 citations

CHARACTERIZATION OF THE k‐SUBTYPE OF THE OPIATE RECEPTOR IN THE GUINEA‐PIG BRAIN

1981 • 423 citations

EFFECTS OF CHANGES IN THE STRUCTURE OF ENKEPHALINS AND OF NARCOTIC ANALGESIC DRUGS ON THEIR INTERACTIONS WITH μ‐ AND δ‐RECEPTORS

1980 • 314 citations

Pharmacological characterization in vivo of the novel opiate, beta-funaltrexamine.

1982 • 296 citations

A novel opioid receptor site directed alkylating agent with irreversible narcotic antagonistic and reversible agonistic activities

1980 • 287 citations

An opioid benzodiazepine

1982 • 201 citations

ASSESSMENT IN THE GUINEA‐PIG ILEUM AND MOUSE VAS DEFERENS OF BENZOMORPHANS WHICH HAVE STRONG ANTINOCICEPTIVE ACTIVITY BUT DO NOT SUBSTITUTE FOR MORPHINE IN THE DEPENDENT MONKEY

1975 • 177 citations

D‐Tyr—Ser—Gly—Phe—Leu—Thr, a highly preferential ligand for δ‐opiate receptors

1980 • 165 citations

COMPARISON OF THE BINDING CHARACTERISTICS OF TRITIATED OPIATES AND OPIOID PEPTIDES

1980 • 155 citations

Opioid binding properties of brain and peripheral tissues: evidence for heterogeneity in opioid ligand binding sites.

1980 • 95 citations

COMPARISON OF THE RECEPTOR BINDING CHARACTERISTICS OF OPIATE AGONISTS INTERACTING WITH μ‐ OR K‐RECEPTORS

1978 • 71 citations

N-[(Tetrahydrofuryl)alkyl] and N-(alkoxyalkyl) derivatives of (-)-normetazocine, compounds with differentiated opioid action profiles

1979 • 69 citations

Improved assays for the assessment of ϰ- and δ-properties of opioid ligands

1982 • 69 citations

Multiplicity of opiate receptors in different species

1982 • 53 citations

Different receptor sites mediate opioid agonism and antagonism

1983 • 43 citations

Profile of activity of κ receptor agonists in the rabbit vas deferens

1985 • 35 citations

Effect of β-FNA on opiate receptor binding: Preliminary evidence for two types of μ receptors

1983 • 34 citations

Studies on the narcotic receptor in the guinea-pig ileum.

1976 • 25 citations

Role of substrate lipophilicity on the N-demethylation and type I binding of 3-O-alkylmorphine analogs

1983 • 14 citations

The binding to rat brain homogenates of Mr2034, a universal opiate

1983 • 10 citations

[3H]tifluadom binding in guinea-pig brain membranes

1984 • 8 citations

Acute and persistent effects of β-funaltrexamine on the binding and agonist potencies of opioids in the myenteric plexus of the guinea-pig ileum

1984 • 6 citations