Identification of a region of the C‐terminal domain involved in short‐term desensitization of the prostaglandin EP₄ receptor

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Cloning, functional expression, and characterization of the human prostaglandin E2 receptor EP2 subtype.

1994 • 244 citations

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Two Gs-coupled prostaglandin E receptor subtypes, EP2 and EP4, differ in desensitization and sensitivity to the metabolic inactivation of the agonist.

1996 • 188 citations

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Two isoforms of prostaglandin E receptor EP3 subtype. Different COOH-terminal domains determine sensitivity to agonist-induced desensitization

1993 • 134 citations

Molecular cloning and expression of multiple isoforms of human prostaglandin E receptor EP3 subtype generated by alternative messenger RNA splicing: multiple second messenger systems and tissue-specific distributions.

1995 • 129 citations

Isoforms of the EP3 Subtype of Human Prostaglandin E2 Receptor Transduce Both Intracellular Calcium and cAMP Signals

1994 • 122 citations

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1994 • 100 citations

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1994 • 85 citations

Molecular Cloning and Expression of Rat Prostaglandin E Receptor EP2 Subtype

1994 • 66 citations

Cloning and expression of a prostaglandin E receptor EP3 subtype from human erythroleukaemia cells

1994 • 65 citations

Selective Regulation of RNK-16 Cell Matrix Metalloproteinases by the EP₄ Subtype of Prostaglandin E₂ Receptor

1996 • 46 citations

The Long Cytoplasmic Carboxyl Terminus of the Prostaglandin E₂Receptor EP₄Subtype Is Essential for Agonist-Induced Desensitization

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Novel mechanism of heterologous desensitization of adenylate cyclase: prostaglandins bind with different affinities to both stimulatory and inhibitory receptors on platelets.

1990 • 30 citations

The C‐terminal domain of the human EP₄ receptor confers agonist‐induced receptor desensitization in a receptor hybrid with the rat EP_3β receptor

1997 • 9 citations