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A common binding site for tricyclic and nontricyclic 5-hydroxytryptamine uptake inhibitors at the substrate recognition site of the neuronal sodium-dependent 5-hydroxytryptamine transporter

Data up to Jan 2025

Published1989
Citations42
References24

Total Citations Per Year

Abstract

References (24)

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1983 • 145 citations

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1985 • 87 citations

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1986 • 80 citations

Differentiation of two components of specific [3H]imipramine binding in rat brain

1984 • 76 citations

High‐ and Low‐Affinity Binding of [3H]Imipramine in Mouse Cerebral Cortex

1983 • 67 citations

Tryptamine, a Substrate for the Serotonin Transporter in Human Platelets, Modifies the Dissociation Kinetics of [3H]Imipramine Binding: Possible Allosteric Interaction

1985 • 65 citations

Serotonin uptake inhibitors differentially modulate high affinity imipramine dissociation in human platelet membranes

1985 • 63 citations

Reaction of the adenine nucleotide analogue 5'-p-fluorosulfonylbenzoyl adenosine at distinct tyrosine and cysteine residues of rabbit muscle pyruvate kinase.

1981 • 58 citations

SL 81.0385: A novel selective and potent serotonin uptake inhibitor

1988 • 42 citations

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1988 • 35 citations

Quantitative Autoradiography of [3H]Indalpine Binding Sites in the Rat Brain: I. Pharmacological Characterization

1985 • 29 citations

High‐ and Low‐Affinity Binding of [3H]Imipramine in Rat Hypothalamus

1986 • 27 citations

Direct and indirect effects of sulfhydryl blocking agents on agonist and antagonist binding to central α1- and α2-adrenoceptors

1984 • 22 citations

Selective effects of thiol reagents on the binding sites for imipramine and neurotransmitter amines in the rat brain

1985 • 21 citations

Chemical modification of α2-adrenoceptors

1986 • 12 citations

Temperature-sensitive conformational changes in [3H]imipramine binding sites and the involvement of sulphur-containing bonds

1984 • 12 citations

Effect of serotonin on the dissociation of high-affinity binding of [3H]imipramine in mouse cerebral cortex

1986 • 8 citations

Evidence for tyrosine at the ligand binding center of beta-adrenergic receptors

1986 • 7 citations

Investigation of membrane located receptors

1985 • 4 citations

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A common binding site for tricyclic and nontricyclic 5-hydroxytryptamine uptake… (1989) – Biochemical Pharmacology | Metascience Observatory Explorer