Molecular aspects of the action of benzodiazepine and nonbenzodiazepine anxiolytics: A hypothetical allosteric model of the benzodiazepine receptor complex

The rat brain: A stereotaxic atlas of the forebrain and lower parts of the brain stem

1986 • 4,155 citations

The pharmacological basis of therapeutics

1981 • 2,853 citations

Benzodiazepine Receptor: Demonstration in the Central Nervous System

1977 • 1,705 citations

Benzodiazepine receptors in rat brain

1977 • 1,459 citations

Specific benzodiazepine receptors in rat brain characterized by high-affinity (3H)diazepam binding.

1977 • 1,246 citations

Amino acid transmitters in the mammalian central nervous system

1974 • 1,169 citations

3H-baclofen and 3H-GABA bind to bicuculline-insensitive GABAB sites in rat brain

1981 • 1,044 citations

GABA‐Benzodiazepine‐Barbiturate Receptor Interactions

1981 • 910 citations

Receptors for the Age of Anxiety: Pharmacology of the Benzodiazepines

1980 • 866 citations

A simple and reliable conflict procedure for testing anti-anxiety agents

1971 • 832 citations

The role of adenosine and its nucleotides in central synaptic transmission

1981 • 767 citations

GABAergic modulation of benzodiazepine binding site sensitivity

1978 • 726 citations

Hypnotics and sedatives

1981 • 712 citations

DRUG INTERACTIONS AT THE GABA RECEPTOR-IONOPHORE COMPLEX

1982 • 696 citations

Adenosine receptors: targets for future drugs

1982 • 681 citations

Isolation, characterization, and purification to homogeneity of an endogenous polypeptide with agonistic action on benzodiazepine receptors.

1983 • 631 citations

Molecular Mechanisms in the Receptor Action of Benzodiazepines

1979 • 579 citations

Diazepam and (--)-pentobarbital: fluctuation analysis reveals different mechanisms for potentiation of gamma-aminobutyric acid responses in cultured central neurons.

1981 • 559 citations

Interaction of Convulsive Ligands with Benzodiazepine Receptors

1982 • 549 citations

Urinary and brain beta-carboline-3-carboxylates as potent inhibitors of brain benzodiazepine receptors.

1980 • 542 citations

New concepts on the mechanism of action of benzodiazepines

1975 • 539 citations

Anticonvulsant activity of (+)‐5‐methyl‐10, 11‐dihydro‐5H‐dibenzo[a, d]cyclohepten‐5, 10‐imine (MK‐801), a substance with potent anticonvulsant, central sympathomimetic, and apparent anxiolytic properties

1982 • 496 citations

An endogenous protein modulates the affinity of GABA and benzodiazepine receptors in rat brain

1978 • 467 citations

The neurobiology of the nucleus accumbens

1982 • 454 citations

Some properties of brain specific benzodiazepine receptors: New evidence for multiple receptors

1979 • 412 citations

Resolution of two biochemically and pharmacologically distinct benzodiazepine receptors

1979 • 408 citations

Characterization of peripheral-type benzodiazepine binding sites in brain using [3H]Ro 5-4864.

1982 • 384 citations

Agonist and antagonist benzodiazepine receptor interaction in vitro

1981 • 383 citations

Radiohistochemical localization of benzodiazepine receptors in rat brain.

1980 • 382 citations

Possible involvement of GABA in the central actions of benzodiazepines.

1975 • 346 citations

Naloxone as a GABA antagonist: Evidence from iontophoretic, receptor binding and convulsant studies

1978 • 330 citations

Molecular heterogeneity of benzodiazepine receptors

1980 • 329 citations

Specific high-affinity binding sites for [3H]Ro 5-4864 in rat brain and kidney.

1983 • 296 citations

Unusual interactions of benzodiazepine receptor antagonists

1982 • 293 citations

A synthetic non-benzodiazepine ligand for benzodiazepine receptors: A probe for investigating neuronal substrates of anxiety

1979 • 284 citations

Benzodiazepines: Potentiation of a GABA inhibitory response in the dorsal raphe nucleus

1978 • 280 citations

Chlordiazepoxide selectively augments GABA action in spinal cord cell cultures

1977 • 280 citations

Benzodiazepine receptor protein identified and visualized in brain tissue by a photoaffinity label.

1980 • 275 citations

Benzodiazepine receptors are coupled to a subpopulation of gamma-aminobutyric acid (GABA) receptors: evidence from a quantitative autoradiographic study.

1981 • 262 citations

Autoradiographic localisation of benzodiazepine receptors in the brains of humans and animals

1979 • 260 citations

[³H]Propyl ?-Carboline-3-Carboxylate as a Selective Radioligand for the BZ₁Benzodiazepine Receptor Subclass

1981 • 255 citations

The effect of diazepam on spinal cord activities: Possible sites and mechanisms of action

1974 • 246 citations

Barbiturate receptor sites are coupled to benzodiazepine receptors.

1980 • 234 citations

Evidence for a late evolutionary appearance of brain-specific benzodiazepine receptors: an investigation of 18 vertebrate and 5 invertebrate species

1978 • 231 citations

Ethyl β-carboline carboxylate lowers seizure threshold and antagonizes flurazepam-induced sedation in rats

1981 • 225 citations

Benzodiazepine Antagonist Ro 15–1788: Binding Characteristics and Interaction with Drug‐Induced Changes in Dopamine Turnover and Cerebellar cGMP Levels

1982 • 222 citations

Stimulation of benzodiazepine receptor binding by gamma-aminobutyric acid.

1979 • 220 citations

Binding of [3H]alpha-dihydropicrotoxinin, a gamma-aminobutyric acid synaptic antagonist, to rat brain membranes.

1978 • 216 citations

Ethyl β-carboline-3-carboxylate shows differential benzodiazepine receptor interaction

1980 • 210 citations

Cyclic Adenosine Monophosphate Phosphodiesterase in Brain: Effect on Anxiety

1972 • 207 citations

Brain Specific Benzodiazepine Receptors

1978 • 205 citations

Is the benzodiazepine receptor coupled to a chloride anion channel?

1979 • 204 citations

An opioid benzodiazepine

1982 • 201 citations

Rapid Changes in Brain Benzodiazepine Receptors After Experimental Seizures

1978 • 196 citations

Purinergic inhibition of diazepam binding to rat brain ()

1979 • 195 citations

β-Carboline-3-carboxylic acid ethyl ester antagonizes diazepam activity

1980 • 193 citations

Purification of an endogenous protein inhibitor of the high affinity binding of gamma-aminobutyric acid to synaptic membranes of rat brain.

1978 • 193 citations

CGS 8216: Receptor binding characteristics of a potent benzodiazepine antagonist

1982 • 192 citations

Nicotinamide is a brain constituent with benzodiazepine-like actions

1979 • 191 citations

Identification of inosine and hypoxanthine as endogenous inhibitors of [3H] diazepam binding in the central nervous system

1978 • 189 citations

.beta.-Carbolines: synthesis and neurochemical and pharmacological actions on brain benzodiazepine receptors

1982 • 175 citations

Anion permeability of the synaptic and non‐synaptic motoneurone membrane

1961 • 171 citations

The effect of γ-aminobutyric acid on 3H-flunitrazepam binding in rat brain

1978 • 170 citations

Relationship between benzodiazepine receptors and experimental anxiety in rats

1978 • 167 citations

Diazepam enhancement of low affinity GABA binding to rat brain membranes

1982 • 166 citations

Identification of inosine and hypoxanthine as endogenous ligands for the brain benzodiazepine-binding sites.

1979 • 166 citations

The proconvulsant and diazepam-reversing effects of ethyl-β-carboline-3-carboxylate

1980 • 162 citations

Die Wirkung von Diazepam auf die pr�synaptische Hemmung und andere R�ckenmarksreflexe

1967 • 156 citations

Effects of two benzodiazepines, phenobarbitone, and baclofen on synaptic transmission in the cat cuneate nucleus

1976 • 155 citations

Micromolar Affinity Benzodiazepine Receptors: Identification and Characterization in Central Nervous System

1982 • 152 citations

Repeated seizures induce long-term increase in hippocampal benzodiazepine receptors.

1980 • 150 citations

Ontogenetic development of benzodiazepine receptors in the rat brain

1978 • 150 citations

Adenosine-dependent formation of cyclic AMP in brain slices

1976 • 149 citations

The Benzodiazepine Receptor in Normal and Pathological Human Brain

1978 • 149 citations

CHARACTERIZATION OF THE BINDING OF [³H]MUSCIMOL, A POTENT γ‐AMINOBUTYRIC ACID AGONIST, TO RAT BRAIN SYNAPTOSOMAL MEMBRANES USING A FILTRATION ASSAY

1979 • 147 citations

Effects of benzodiazepines on central serotonergic mechanisms.

1975 • 143 citations

Evidence for involvement of GABA in the action of benzodiazepines: studies on rat cerebellum.

1975 • 141 citations

[3H]Diazepam binding in mammalian central nervous system: a pharmacological characterization

1981 • 141 citations

Buspirone: Effects on central monoaminergic transmission - possible relevance to animal experimental and clinical findings

1982 • 139 citations

Restoration of shock‐suppressed behavior by treatment with (+)‐5‐methyl‐10,11‐dihydro‐5H‐dibenzo[a, d]cyclohepten‐5, 10‐imine (MK‐801), a substance with potent anticonvulsant, central sympathomimetic, and apparent anxiolytic properties

1982 • 137 citations

Is stimulation of benzodiazepine receptor binding mediated by a novel GABA receptor?

1979 • 135 citations

Buspirone: Action on serotonin receptors in calf hippocampus

1983 • 127 citations

Cellular Mechanisms of Benzodiazepine Action

1982 • 127 citations

Correlation between benzodiazepine receptor occupation and anticonvulsant effects of diazepam

1979 • 127 citations

GABA reduces binding of 3H-methyl β-carboline-3-carboxylate to brain benzodiazepine receptors

1981 • 126 citations

Ontogeny of GABA and benzodiazepine receptors: Effects of Triton X-100, bromide and muscimol

1979 • 124 citations

The effects of naloxone and picrotoxin on the sedative and anticonflict effects of benzodiazepines

1978 • 124 citations

Pharmacology of the benzodiazepines

1985 • 120 citations

Multiple benzodiazepine receptors: Evidence of a dissociation between anticonflict and anticonvulsant properties by PK 8165 and PK 9084 (two quinoline derivatives)

1981 • 120 citations

The mechanism(s) of action of the benzodiazepines

1981 • 117 citations

and inhibition by zopiclone of benzodiazepine binding to rodent brain receptors

1979 • 117 citations

Benzodiazepine Inhibition of the Calcium-Calmodulin Protein Kinase System in Brain Membrane

1981 • 115 citations

Dopamine and antianxiety activity

1982 • 114 citations

No changes in rat benzodiazepine receptors after withdrawal from continuous treatment with lorazepam and diazepam

1979 • 110 citations

Neurotransmitter receptor localizations: Brain lesion induced alterations in benzodiazepine, GABA, β-adrenergic and histamine H1-receptor binding

1980 • 108 citations

Benzodiazepine binding sites: receptors or acceptors?

1982 • 108 citations

Peripheral benzodiazepine binding sites in heart and their interaction with dipyridamole

1981 • 108 citations

Enhancement of the binding of 3H-diazepam to rat brain membranes by SQ 20009, a novel anxiolytic, γ-aminobutyric acid (GABA) and muscimol

1979 • 106 citations

gamma-Aminobutyric acid and benzodiazepine receptors: copurification and characterization.

1981 • 105 citations

Molecular substrates of anxiety: Clues from the heterogeneity of benzodiazepine receptors

1982 • 105 citations

The Binding of the GAB A Agonist [³H]THIP to Rat Brain Synaptic Membranes

1982 • 102 citations

The anionic permeability of the inhibitory postsynaptic membrane of hippocampal pyramidal cells

1977 • 101 citations

Solubilization of histamine H-1, GABA and benzodiazepine receptors

1979 • 99 citations

Biochemical identification of pharmacologically and functionally distinct GABA receptors in rat brain

1981 • 97 citations

Characterization of photoaffinity labeling of benzodiazepine binding sites.

1981 • 95 citations

Enhancement of benzodiazepine and GABA binding by the novel anxiolytic, tracazolate

1982 • 93 citations

Chronic clonazepam administration induced benzodiazepine receptor subsensitivity

1982 • 91 citations

Inhibition of diazepam binding by tryptophan derivatives including melatonin and its brain metabolite N-acetyl-5-methoxy kynurenamine

1981 • 91 citations

Physical separation and characterization of two types of benzodiazepine receptors.

1982 • 90 citations

[³H]Propyl ?-Carboline-3-Carboxylate Binds Specifically to Brain Benzodiazepine Receptors

1981 • 89 citations

Characterization of benzodiazepine and gamma-aminobutyric recognition sites and their endogenous modulators

1981 • 89 citations

A steroid derivative, R 5135, antagonizes the GABA/benzodiazepine receptor interaction

1981 • 88 citations

Perturbation of benzodiazepine receptor binding by pyrazolopyridines involves picrotoxinin/barbiturate receptor sites

1981 • 82 citations

GABA binding in mammalian brain: Inhibition by endogenous GABA

1980 • 81 citations

Enhancement of 3H-diazepam binding by SQ 65,396: A novel anti-anxiety agent

1978 • 80 citations

In vitro modulations by SQ 20009 and SQ 65396 of GABA receptor binding in rat CNS membranes

1980 • 80 citations

Solubilization of benzodiazepine binding site from rat cortex

1979 • 78 citations

Benzodiazepine receptors: Differential interaction of benzodiazepine agonists and antagonists after photoaffinity labeling with flunitrazepam

1982 • 78 citations

Benzodiazepines: GABA and glycine receptors on single neurons in the rat medulla

1976 • 78 citations

Multiple benzodiazepine receptors and their regulation by γ-aminobutyric

1981 • 77 citations

Ontogenetic changes in GABA modulation of brain benzodiazepine binding

1980 • 76 citations

Avermectin B_1a Modulation of γ‐Aminobutyric Acid Receptors in Rat Brain Membranes

1982 • 76 citations

Interactions of barbiturates of various pharmacological categories with benzodiazepine receptors.

1982 • 75 citations

Diazepam and presynaptic inhibition

1971 • 74 citations

Inosine, an endogenous ligand of the brain benzodiazepine receptor, antagonizes pentylenetetrazole-evoked seizures.

1979 • 73 citations

Methyl-β-carboline-induced convulsions are antagonized by Ro 15-1788 and by propyl-β-carboline

1982 • 71 citations

Some properties of 3H-diazepam displacing activity from human urine

1979 • 70 citations

Multiple benzodiazepine receptors: Structures in the brain or structures in the mind? A critical review

1983 • 68 citations

Demonstration of an endogenous, competitive inhibitor(s) of [3H] diazepam binding in bovine brain

1978 • 66 citations

Mechanism of action of the benzodiazepines: behavioral aspect.

1980 • 66 citations

Heterogeneity of benzodiazepine receptor interactions with gamma-aminobutyric acid and barbiturate receptor sites.

1983 • 66 citations

The role of GABA in mediating the anticonvulsant properties of benzodiazepines

1980 • 65 citations

Buspirone enhances [3H]flunitrazepam binding in vivo

1983 • 65 citations

Evidence that benzodiazepine receptors reside on cerebellar purkinje cells: Studies with “nervous” mutant mice

1978 • 64 citations

Interaction of diphenylhydantoin and benzodiazepines in the CNS

1980 • 63 citations

Displacement of [3H] diazepam binding in rat brain by dipyridamole and by 1-methylisoguanosine, a marine natural product with muscle relaxant activity

1980 • 63 citations

Enhancement of in vitro binding and some of the pharmacological properties of diazepam by a novel anthelmintic agent, avermectin B1a

1979 • 62 citations

Pentobarbital potentiates GABA-enhanced [3H]-diazepam binding to benzodiazepine receptors

1980 • 62 citations

Identification of an endogenous peptide-ligand for the benzodiazepine receptor

1980 • 62 citations

Stimulation of benzodiazepine receptor binding by SQ 20009 is chloride-dependent and picrotoxin-sensitive

1979 • 59 citations

Reduction in benzodiazepine receptors associated with Purkinje cell degeneration in ‘nervous’ mutant mice

1979 • 59 citations

Studies on the relationship of gamma-aminobutyric acid-stimulated diazepam binding and the gamma-aminobutyric acid receptor.

1981 • 59 citations

Suriclone: A New Cyclopyrrolone Derivative Recognizing Receptors Labeled by Benzodiazepines in Rat Hippocampus and Cerebellum

1983 • 58 citations

Enhancement by anesthetic and convulsant barbiturates of GABA binding to rat brain synaptosomal membranes

1981 • 58 citations

Anxioselective anxiolytics

1983 • 56 citations

Soluble benzodiazepine receptors: Gabaergic regulation

1980 • 55 citations

Competitive inhibition of benzodiazepine binding by fractions from porcine brain.

1978 • 55 citations

Analgesic Action and Pharmacokinetics of Morphine and Diazepam in Man

1979 • 55 citations

[Effect of diazepam on presynaptic inhibition and other spinal reflexes].

1967 • 54 citations

Heterogeneity of Benzodiazepine Receptors in the Central Nervous System Demonstrated with Kenazepine, an Alkylating Benzodiazepine

1980 • 53 citations

Dihydropicrotoxinin binding sites in mammalian brain: Interaction with convulsant and depressant benzodiazepines

1981 • 51 citations

Modulation of benzodiazepine receptor binding: Insight into pharmacological efficacy

1982 • 51 citations

Modulation by picrotoxin and IPTBO of 3H-flunitrazepam binding to the GABA/benzodiazepine receptor complex of rat cerebellum

1981 • 50 citations

Interaction of putative anxiolytic agents with central adenosine receptors

1981 • 49 citations

Heterogeneity of brain benzodiazepine receptors demonstrated by [3H]propyl beta-carboline-3-carboxylate binding.

1982 • 47 citations

Antagonistic action of diphenylhydantoin and calcium on the level of phosphorylation of particular rat and human brain proteins

1977 • 47 citations

Binding of a radiolabeled triazolopyridazine to a subtype of benzodiazepine receptor in the rat cerebellum.

1982 • 46 citations

Effects of naloxone on the anticonflict properties of alcohol and chlordiazepoxide.

1980 • 46 citations

Molecular size of benzodiazepine receptor in rat brain in situ: evidence for a functional dimer?

1982 • 44 citations

Solubilization and properties of a benzodiazepine receptor from calf cortex

1980 • 43 citations

Interaction of SQ 20009 and GABA-like drugs as modulators of benzodiazepine receptor binding

1980 • 43 citations

Chronic benzodiazepine treatment increases [3H]muscimol binding in mouse brain

1982 • 43 citations

Photoaffinity labeling of benzodiazepine receptors causes altered agonist-antagonist interactions

1983 • 41 citations

γ-Aminobutyric acid regulation of the benzodiazepine receptor: biochemical evidence for pharmacologically different effects of benzodiazepines and propyl β-carboline-3-carboxylate

1981 • 41 citations

Interactions between narcotic analgesics and benzodiazepine derivatives on behavior in the mouse.

1976 • 41 citations

Demonstration of brain-specific benzodiazepine receptors in rat retina

1980 • 40 citations

Avermectin B1a: An irreversible activator of the γ-aminobutyric acid-benzodiazepine-chloride-ionophore receptor complex

1980 • 40 citations

Kinetics of [3H]flunitrazepam binding to membrane-bound benzodiazepine receptors.

1982 • 40 citations

Anxiolytic Properties of Opiates and Endogenous Opioid Peptides and Their Relationship to the Actions of Benzodiazepines1

2015 • 40 citations

Searching for endogenous benzodiazepine receptor ligands

1980 • 40 citations

Endogenous effector of the benzodiazepine binding site: purification and characterization

1981 • 40 citations

A study of the influence of hydroxyzine and diazepam on morphine antinociception in the rat

1979 • 39 citations

The inhibition of GABA-stimulated benzodiazepine binding by a convulsant benzodiazepine

1980 • 38 citations

Facilitation of specific benzodiazepine binding in rat brain membrane fragments by a number of anions

1980 • 38 citations

In Vitro Modulation by Avermectin B₁a of the GABA/Benzodiazepine Receptor Complex of Rat Cerebellum

1981 • 37 citations

Action of the benzodiazepines on the cholinergic system.

1975 • 37 citations

Thromboxane A2 as a possible natural ligand for benzodiazepine receptors

1978 • 37 citations

Benzodiazepines and neurotransmitters.

1980 • 36 citations

GABA-benzodiazepine interactions: physiological, pharmacological and developmental aspects.

1980 • 36 citations

A comparative study of avermectin B1a and other modulators of the gamma- aminobutyric acid receptor . chloride ion channel complex

1982 • 35 citations

Thyroid Hormones and Derivatives Inhibit Flunitrazepam Binding

1983 • 34 citations

Effects of Cations and Anions on the Binding of 3H-Diazepam to Rat Brain

1978 • 34 citations

Acute diazepam administration produces rapid increases in brain benzodiazepine receptor density

1979 • 34 citations

Benzodiazepine receptors: Alterations in mutant mouse cerebellum

1979 • 34 citations

Evidence that ethanol and pentobarbital enhance [3h]diazepam binding at the benzodiazepine-GABA receptor-ionophore complex indirectly

1981 • 34 citations

Inhibition of [³H]Diazepam and [³H]3‐Carboethoxy‐β‐Carboline Binding by Irazepine: Evidence for Multiple “Domains” of the Benzodiazepine Receptor

1982 • 32 citations

Electrophysiological actions of benzodiazepines.

1980 • 31 citations

The Relationship of Anxiety to Depression

1982 • 31 citations

Photoaffinity labelling of the benzodiazepine receptor cannot be used to predict ligand efficacy

1983 • 30 citations

Modulation of benzodiazepine binding site sensitivity

1979 • 30 citations

Pharmacologic and behavioral effects of EMD 28422: A novel purine which enhances (3H) diazepam binding to brain benzodiazepine receptors

1980 • 30 citations

Purine inhibition of [3H]-γ-aminobutyric acid receptor binding to rat brain membranes

1980 • 30 citations

Benzodiazepines are weak inhibitors of [3H]nitrobenzylthioinosine binding to adenosine uptake sites in brain

1982 • 30 citations

Effect of the benzodiazepine receptor antagonist Ro 15-1788 on the anticonvulsant and anticonflict actions of MK-801

1982 • 30 citations

The role of central glycine receptors in the pharmacologic actions of benzodiazepines.

1975 • 29 citations

GABA and barbiturate receptors

1982 • 28 citations

Buspirone analogs. 1. Structure-activity relationships in a series of N-aryl- and heteroarylpiperazine derivatives

1983 • 28 citations

Differential effects of Triton X-100 on benzodiazepine and GABA binding in a frozen-thawed synaptosomal fraction of rat brain

1979 • 25 citations

Contrasting regulation by GABA of the displacement of benzodiazepine antagonist binding by benzodiazepine agonists and purines

1982 • 25 citations

Stimulation of benzodiazepine binding to rat brain membranes and solubilized receptor complex by avermectin B1a and γ-aminobutyric acid

1981 • 25 citations

GABA receptors regulate the affinities of anions required for brain specific benzodiazepine binding.

1981 • 24 citations

Ivermectin Interactions with Benzodiazepine Receptors in Rat Cortex and Cerebellum In Vitro

1984 • 24 citations

Comparative Thermodynamics of Benzodiazepine Receptor Ligand Interactions in Rat Neuronal Membranes

1983 • 24 citations

Increased benzodiazepine receptor number elicited in vitro by a novel purine, EMD 28422

1980 • 24 citations

Inhibition of γ-aminobutyric acid stimulated [3H]diazepam binding by benzodiazepine receptor ligands

1981 • 23 citations

Etazolate (SQ20009): electrophysiology and effects on [3H]flunitrazepam binding in cultured cortical neurons

1983 • 23 citations

[3H]ethyl β-carboline-3-carboxylate binding to the benzodiazepine receptors is not affected by GABA

1981 • 22 citations

Inhibition by etazolate (SQ 20009) and cartazolate (SQ 65396) of adenosine-stimulated [3H]cAMP formation in [2-3H]adenine-prelabeled vesicles prepared from guinea pig cerebral cortex

1982 • 22 citations

Influence of morphine dependence on GABA-stimulated benzodiazepine binding to mouse brain synaptic membranes

1982 • 22 citations

?-Carboline binding indicates the presence of benzodiazepine receptor subclasses in the bovine central nervous system

1982 • 22 citations

Competition for diazepam receptor binding by diphenylhydantoin and its enhancement by γ-aminobutyric acid

1979 • 22 citations

The Benzodiazepine Receptor in Rat Brain and Its Interaction with Ethyl /3‐Carboline‐3‐Carboxylate

1983 • 21 citations

Prostaglandins a as possible endogenous ligands of benzodiazepine receptor

1982 • 20 citations

Interaction of avermectins with [3H]β-carboline-3-carboxylate ethyl ester and [3H]Diazepam binding sites in rat brain cortical membranes

1982 • 19 citations

Changes in mouse brain diazepam receptor binding after phenobarbital administration

1980 • 19 citations

The effect of GABA on binding of two novel non-benzodiazepines, PK 8165 and CGS 8216, to benzodiazepine receptors in the rat brain

1982 • 18 citations

CGS 7525A, A new, centrally active alpha2 adrenoceptor antagonist

1983 • 17 citations

Two or more conformations of benzodiazepine receptors depending on GABA receptors and other variables.

1980 • 17 citations

Interaction of the benzodiazepine antagonists, CGS 8216 and Ro 15-1788, with central adenosine A-1 receptors.

1982 • 16 citations

Molecular Interactions of Etazolate with Benzodiazepine and Picrotoxinin Binding Sites

1982 • 14 citations

Problems in the electrophysiological analysis of the site of action of benzodiazepines.

1975 • 13 citations

Pharmacodynamic effects and possible therapeutic uses of THIP, a specific GABA-agonist

1982 • 12 citations

U 43,465F: A benzodiazepine with antidepressant activity? interaction with Ro 15–1788 and d,l-propranolol

1982 • 12 citations

Evidence for GABA involvement in the action of diazepam on presynaptic nerve terminals in bullfrog sympathetic ganglia.

1975 • 11 citations

[3H] Diazepam Displacing Activity in Human Cerebrospinal Fluid

1981 • 11 citations

GABA and benzodiazepine receptors. Studies on their localization in the hippocampus and their interaction with central dopamine neurons in the rat brain.

1981 • 11 citations

Ineffectiveness of a purine analogue, EMD 28422, in two animal tests of anxiolytic action

1983 • 10 citations

High affinity inhibition of [3H]-Flunitrazepam binding to brain benzodiazepine receptors by CGS 9896, a novel pyrazoloquinoline

1982 • 10 citations

Lateral olfactory tract lesions reveal neuronal localization of benzodiazepine recognition sites

1981 • 8 citations

Studies on benzodiazepine receptors.

1980 • 8 citations

Antagonism of the anxiolytic action of diazepam and chlordiazepoxide by the novel imidazopyridines, EMD 39593 and EMD 41717

1983 • 8 citations

Pharmacological and biochemical evidence for an interaction between the benzodiazepine and GABA receptors.

1980 • 7 citations

Glycine, GABA and Benzodiazepine Receptors

1980 • 6 citations

Inactivation of GABA receptors by phenoxybenzamine: Effects on GABA-stimulated benzodiazepine binding in the central nervous system

1982 • 5 citations

Neurotransmitter Receptors, Part I: Amino Acids, Peptides and Benzodiazepines

1981 • 5 citations

Animal psychopharmacological models: Use of conflict behavior in predicting clinical effects of anxiolytics and their mechanism of action

1982 • 4 citations

Demonstration and characterization of an endogenous inhibitor of GABA-enhanced [3H]-diazepam binding from bovine cerebral cortex.

1981 • 4 citations

Effect of benzodiazepines on the central action of narcotic analgesics.

1982 • 4 citations