Tissue Distribution, Autoradiography, and Metabolism of 4‐(2′‐Methoxyphenyl)‐1‐[2′ ‐[N‐2″‐Pyridinyl)‐p‐[¹⁸F]Fluorobenzamido]ethyl]piperazine (p‐[¹⁸F]MPPF), a New Serotonin 5‐HT_1A Antagonist for Positron Emission Tomography

Identification of presynaptic serotonin autoreceptors using a new ligand: 3H-PAT

1983 • 759 citations

A pharmacological profile of the selective silent 5-HT1A receptor antagonist, WAY-100635

1995 • 610 citations

Electrophysiological, biochemical, neurohormonal and behavioural studies with WAY-100635, a potent, selective and silent 5-HT1A receptor antagonist

1995 • 515 citations

Quantitative autoradiography of multiple 5-HT1 receptor subtypes in the brain of control or 5,7-dihydroxytryptamine-treated rats

1986 • 513 citations

The concept of selectivity in 5-HT receptor research

1990 • 425 citations

Immunocytochemical localization of serotonin1A receptors in the rat central nervous system

1996 • 370 citations

Exquisite delineation of 5-HT1A receptors in human brain with PET and [carbonyl-11C]WAY-100635

1996 • 226 citations

Serotonin receptors: Subtypes, functional responses and therapeutic relevance

1995 • 224 citations

Evidence for the localization of 5HT1A binding sites on serotonin containing neurons in the raphe dorsalis and raphe centralis nuclei of the rat brain

1985 • 202 citations

Serotonin receptors: Clinical implications

1990 • 196 citations

5-Hydroxytryptamine receptor subtypes in vertebrates and invertebrates

1994 • 182 citations

The selective 5-HT1A antagonist radioligand [3H]WAY 100635 labels both G-protein-coupled and free 5-HT1A receptors in rat brain membranes

1995 • 178 citations

Fluorine-18-altanserin: a radioligand for the study of serotonin receptors with PET: radiolabeling and in vivo biologic behavior in rats.

1991 • 167 citations

Effects of acute fluoxetine on extracellular serotonin levels in the raphe: an in vivo microdialysis study

1995 • 157 citations

Serotonin Receptor Subtypes

1995 • 149 citations

High-Yield Radiosynthesis and Preliminary In Vivo Evaluation of p-[18F]MPPF, a Fluoro Analog of WAY-100635

1998 • 139 citations

Effect of fluoxetine on extracellular 5-hydroxytryptamine in rat brain. Role of 5-HT autoreceptors

1998 • 118 citations

Quantitative autoradiographic characterisation of the binding of [3H]WAY-100635, a selective 5-HT1A receptor antagonist

1995 • 113 citations

Synthesis And Evaluation of 4-(2'-Methoxyphenyl)-1-[2'-[N-(2''-pyridinyl)- p-iodobenzamido]ethyl]piperazine (p-MPPI): A New Iodinated 5-HT1A Ligand

1994 • 107 citations

Selective in vivo labelling of brain 5-HT1A receptors by [3H]WAY 100635 in the mouse

1994 • 106 citations

p-[18F]-MPPF: A potential radioligand for PET studies of 5-HT1A receptors in humans

1997 • 102 citations

The Main Features of Central 5-HT1A Receptors

2000 • 98 citations

5-HT receptor subtypes outside the central nervous system. Roles in the physiology of the gut.

1990 • 90 citations

Effects of Sleep Deprivation on Serotonergic Neuronal Activity in the Dorsal Raphe Nucleus of the Freely Moving Cat

1997 • 89 citations

Evidence for 5‐HT₁‐like receptor‐mediated vasoconstriction in human pulmonary artery

1996 • 87 citations

The main features of central 5-HT1 receptors.

1989 • 55 citations

Short Communication New 5-HT1A receptor antagonist: [3H]p-MPPF

1996 • 55 citations

4-(2'-Methoxyphenyl)-1-[2'-[N-(2"-pyridinyl)-p-iodobenzamido]ethyl] piperazine and 4-(2'-methoxyphenyl)-1-[2'-[N-(2"-pyridinyl)-p- fluorobenzamido]ethyl]piperazine, two new antagonists at pre- and postsynaptic serotonin-1A receptors.

1996 • 46 citations

Mitogenic effect of serotonin in human small cell lung carcinoma cells via both 5-HT1A and 5-HT1D receptors

1995 • 45 citations

A chronic arterial and venous cannulation method for freely moving rats

1985 • 39 citations

In vivo characterization of p-[18F]MPPF, a fluoro analog of WAY-100635 for visualization of 5-HT1a receptors

2000 • 37 citations

Human sleep EEG following the 5-HT1A antagonist pindolol: possible disinhibition of raphe neuron activity

1997 • 28 citations

Role of 5‐HT_1A Receptors in Acquisition, Consolidation and Retrieval of Learning

1997 • 23 citations

Robot-assisted synthesis of [18F]altanserin, 4-[18F]fluorotropapride, 6-[18F]fluoro-L-dopa and 2-[18F]fluoro-L-tyrosine.

1994 • 3 citations