[³H]‐L‐2‐amino‐4‐phosphonobutyrate labels a metabotropic glutamate receptor, mGluR4a

The Excitatory Amino Acid Receptors: Their Classes, Pharmacology, and Distinct Properties in the Function of the Central Nervous System

1989 • 2,203 citations

MODEL SYSTEMS FOR THE STUDY OF SEVEN-TRANSMEMBRANE-SEGMENT RECEPTORS

1991 • 1,357 citations

Muscarinic Receptors—Characterization, coupling and function

1993 • 1,264 citations

Molecular characterization of a novel retinal metabotropic glutamate receptor mGluR6 with a high agonist selectivity for L-2-amino-4-phosphonobutyrate

1993 • 724 citations

The ligand-binding domain in metabotropic glutamate receptors is related to bacterial periplasmic binding proteins

1993 • 695 citations

Signal transduction, pharmacological properties, and expression patterns of two rat metabotropic glutamate receptors, mGluR3 and mGluR4

1993 • 585 citations

Molecular characterization of a new metabotropic glutamate receptor mGluR7 coupled to inhibitory cyclic AMP signal transduction.

1994 • 466 citations

A novel metabotropic glutamate receptor expressed in the retina and olfactory bulb

1995 • 328 citations

Analysis of agonist and antagonist activities of phenylglycine derivatives for different cloned metabotropic glutamate receptor subtypes

1994 • 323 citations

Micromolar L-2-amino-4-phosphonobutyric acid selectively inhibits perforant path synapses from lateral entorhinal cortex

1981 • 307 citations

Presynaptic glutamate receptors depress excitatory monosynaptic transmission between mouse hippocampal neurones.

1990 • 249 citations

Cloning and expression of a new member of the L-2-amino-4-phosphonobutyric acid-sensitive class of metabotropic glutamate receptors.

1994 • 246 citations

Cloning and expression of an A1 adenosine receptor from rat brain.

1991 • 235 citations

Partial agonists, full agonists, antagonists: dilemmas of definition

1993 • 234 citations

Domains involved in the specificity of G protein activation in phospholipase C-coupled metabotropic glutamate receptors.

1994 • 197 citations

Agonist analysis of 2‐(carboxycyclopropyl)glycine isomers for cloned metabotropic glutamate receptor subtypes expressed in Chinese hamster ovary cells

1992 • 189 citations

The Ca²⁺/Cl⁻ dependent L‐[³H]glutamate binding: a new receptor or a particular transport process?

1984 • 169 citations

Actions of phenylglycine analogs at subtypes of the metabotropic glutamate receptor family

1994 • 139 citations

L-2-amino-4-phosphonobutyrate (L-AP4) is an agonist at the type iv metabotropic glutamate receptor which is negatively coupled to adenylate cyclase

1992 • 135 citations

Species difference in the G protein selectivity of the human and bovine A1-adenosine receptor.

1994 • 113 citations

Trans-ACPD and l-APB presynaptically inhibit excitatory glutamatergic transmission in the basolateral amygdala (BLA)

1992 • 80 citations

Synthesis of [3H]2-Amino-4-phosphonobutyric acid and characterization of its binding to rat brain membranes: a selective ligand for the chloride/calcium-dependent class ofl-glutamate binding sites

1983 • 74 citations

Characterization of the binding of <scp>dl</scp>‐[³H]‐2‐amino‐4‐phosphonobutyrate to <scp>l</scp>‐glutamate‐sensitive sites on rat brain synaptic membranes

1983 • 62 citations

Characteristics of chloride-dependent incorporation of glutamate into brain membranes argue against a receptor binding site

1987 • 60 citations

<scp>l</scp>‐Glutamate Uptake Inhibitors May Stimulate Phosphoinositide Hydrolysis in Baby Hamster Kidney Cells Expressing mGluR1a via Heteroexchange with <scp>l</scp>‐Glutamate Without Direct Activation of mGluR1a

1994 • 60 citations

Expression pattern and pharmacology of the rat type IV metabotropic glutamate receptor

1993 • 56 citations

Cl⁻/Ca²⁺‐dependent L‐glutamate binding sites do not correspond to 2‐amino‐4‐phosphonobutanoate‐sensitive excitatory amino acid receptors

1985 • 52 citations

Excitatory amino acid receptors — Design of agonists and antagonists

1993 • 50 citations

Metabotropic glutamate receptor heterogeneity in rat brain.

1994 • 46 citations

1S,3R-ACPD-sensitive (metabotropic) [3H]glutamate receptor binding in membranes

1992 • 43 citations

Cyclic analogs of 2-amino-4-phosphonobutanoic acid (APB) and their inhibition of hippocampal excitatory transmission and displacement of [3H]APB binding

1986 • 37 citations

Molecular Cloning, Expression, and Characterization of Metabotropic Glutamate Receptor Subtypes

1994 • 33 citations

Chloride transport blockers inhibit the chloride-dependent glutamate binding to rat brain membranes

1987 • 33 citations

Serine-O-phosphate has affinity for type IV, but not type I, metabotropic glutamate receptor.

1993 • 30 citations

Stimulation intensity as critical determinant of presynaptic receptor effectiveness

1990 • 29 citations

Displacement of DL-[3H]-2-amino-4-phosphonobutanoic acid ([3H]APB) binding with methyl-substituted APB analogs and glutamate agonists

1985 • 27 citations

L-2-amino-4-phosphonobutanoic acid and 1S,3R-1-aminocyclopentane-1,3-dicarboxylic acid reduce paired-pulse depression recorded from medial perforant path in the dentate gyrus of rat hippocampal slices.

1993 • 19 citations

Antioxidant protection of Bio-normalizer in cerebral ischaemia-reperfusion injury in the gerbil

1993 • 16 citations

Activity of the conformationally rigid 2-amino-4-phosphonobutanoic acid (AP4) analogue (RS)-1-amino-3-(phosphonomethylene)cyclobutane-1-carboxyclic acid (cyclobutylene AP5) on evoked responses in the perforant pathway of rat hippocampus

1992 • 12 citations

dl-2-[3,4-3H]Amino-4-phosphonobutyrate binding sites in the rat hippocampus: distribution and possible physiological role

1987 • 12 citations

Effects of bromohomoibotenate on metabotropic glutamate receptors

1994 • 9 citations