Back to search

Delta opioid receptor down-regulation is independent of functional G protein yet is dependent on agonist efficacy.

Data up to Jan 2025

Published1998
Citations22
References28

Total Citations Per Year

Abstract

References (28)

PROTEIN MEASUREMENT WITH THE FOLIN PHENOL REAGENT

1951 • 319,299 citations

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1973 • 12,522 citations

Cloning of a Delta Opioid Receptor by Functional Expression

1992 • 1,225 citations

CLASSIFICATION OF OPIOID RECEPTORS

1983 • 787 citations

International Union of Pharmacology. XII. Classification of opioid receptors.

1996 • 704 citations

Dimerization of the δ Opioid Receptor:

1997 • 479 citations

Under Siege: The Brain on Opiates

1996 • 263 citations

μ Opioid Receptor Phosphorylation, Desensitization, and Ligand Efficacy

1997 • 218 citations

Sequestration of the δ Opioid Receptor

1996 • 198 citations

Characterization of opioid agonist efficacy in a C6 glioma cell line expressing the mu opioid receptor.

1996 • 173 citations

Adenylylcyclase Supersensitization in μ-Opioid Receptor-transfected Chinese Hamster Ovary Cells Following Chronic Opioid Treatment

1995 • 162 citations

Visualization of Agonist-induced Sequestration and Down-regulation of a Green Fluorescent Protein-tagged β2-Adrenergic Receptor

1998 • 158 citations

Determinants of alpha 2-adrenergic receptor activation of G proteins: evidence for a precoupled receptor/G protein state.

1994 • 149 citations

Inhibition of the ω-conotoxin-sensitive calcium current by distinct G proteins

1992 • 128 citations

Regulation of Multiple Effectors by the Cloned δ‐Opioid Receptor: Stimulation of Phospholipase C and Type II Adenylyl Cyclase

1995 • 116 citations

Go mediates the coupling of the mu opioid receptor to adenylyl cyclase in cloned neural cells and brain.

1993 • 111 citations

beta-Adrenergic receptor kinase. Activity of partial agonists for stimulation of adenylate cyclase correlates with ability to promote receptor phosphorylation.

1988 • 106 citations

Thr353, Located within the COOH-terminal Tail of the ´ Opiate Receptor, Is Involved in Receptor Down-regulation

1996 • 105 citations

A Chimeric Study of the Molecular Basis of Affinity and Selectivity of the κ and the δ Opioid Receptors.

1995 • 98 citations

Down-regulation of μ-Opioid Receptor by Full but Not Partial Agonists Is Independent of G Protein Coupling

1997 • 78 citations

The μ-Opioid Receptor Down-Regulates Differently from the δ-Opioid Receptor: Requirement of a High Affinity Receptor/G Protein Complex Formation

1997 • 72 citations

Acute and Chronic Effects of Opioids on δ and μ Receptor Activation of G Proteins in NG108‐15 and SK‐N‐SH Cell Membranes

1997 • 64 citations

Opioid efficacy in a C6 glioma cell line stably expressing the delta opioid receptor.

1997 • 56 citations

SCATCHARD ANALYSIS OF OPIATE RECEPTOR BINDING

1980 • 41 citations

beta-Adrenergic-receptor kinase

1997 • 37 citations

Opioid Regulation of the Mouse δ-Opioid Receptor Expressed in Human Embryonic Kidney 293 Cells

1997 • 37 citations

The Involvement of Novel Protein Kinase C Isozymes in Influencing Sensitivity of Breast Cancer MCF-7 Cells to Tumor Necrosis Factor-α

1998 • 37 citations

Opiate Receptor Changes after Chronic Exposure to Agonists and Antagonists

1995 • 36 citations

Cited By (0)

Loading...
Delta opioid receptor down-regulation is independent of functional G protein yet is… (1998) – PubMed | Metascience Observatory Explorer