5‐HT₃ Receptors

Proposals for the classification and nomenclature of functional receptors for 5-hydroxytryptamine

1986 • 1,255 citations

Identification and distribution of 5-HT3 receptors in rat brain using radioligand binding

1987 • 866 citations

Identification of serotonin M-receptor subtypes and their specific blockade by a new class of drugs

1985 • 845 citations

TWO KINDS OF TRYPTAMINE RECEPTOR

1957 • 838 citations

Identity of inhibitory presynaptic 5-hydroxytryptamine (5-HT) autoreceptors in the rat brain cortex with 5-HT1B binding sites

1986 • 686 citations

5-HT3 receptors are membrane ion channels

1989 • 630 citations

Pharmacological properties of GR38032F, a novel antagonist at 5‐HT₃ receptors

1988 • 378 citations

Effects of the 5‐HT₃ receptor antagonist, GR38032F, on raised dopaminergic activity in the mesolimbic system of the rat and marmoset brain

1987 • 354 citations

Inhibition of cisplatin‐induced vomiting by selective 5‐hydroxytryptamine M‐receptor antagonism

1986 • 336 citations

Differential inhibitory effects of a 5-HT3 antagonist on drug-induced stimulation of dopamine release

1989 • 277 citations

Pharmacological characterization of 5‐hydroxytryptamine‐induced depolarization of the rat isolated vagus nerve

1987 • 276 citations

5-HT3 receptors mediate inhibition of acetylcholine release in cortical tissue

1989 • 259 citations

Binding of the 5-HT3 ligand, [3H]GR65630, to rat area postrema, vagus nerve and the brains of several species

1989 • 230 citations

5‐HT₃ receptor antagonists injected into the area postrema inhibit cisplatin‐induced emesis in the ferret

1989 • 218 citations

Selective and functional 5-hydroxytryptamine3 receptor antagonism by BRL 43694 (granisetron)

1989 • 216 citations

Pharmacological analysis of drug-receptor interaction

1994 • 212 citations

Action of drugs of abuse on brain reward systems: An update with specific attention to opiates

1982 • 194 citations

Study of the contractile effect of 5-hydroxytryptamine (5-HT) in the isolated longitudinal muscle strip from guinea-pig ileum

1985 • 194 citations

PREVENTION OF EMESIS IN PATIENTS RECEIVING CYTOTOXIC DRUGS BY GR38032F, A SELECTIVE 5-HT3 RECEPTOR ANTAGONIST

1987 • 193 citations

5-hydroxytryptamine m-receptor antagonism to prevent cisplatin-induced emesis

1986 • 190 citations

5-HT3 receptor binding sites are on capsaicin-sensitive fibres in the rat spinal cord

1989 • 184 citations

5HT3 receptor antagonists block morphine- and nicotine-but not amphetamine-induced reward

1989 • 176 citations

Effects of capsaicin on nociceptive heat, pressure and chemical thresholds and on substance P levels in the rat

1980 • 167 citations

Localisation by autoradiography of neuronal 5-HT3 receptors in the mouse CNS

1988 • 164 citations

Activation of a 5-HT3 receptor releases dopamine from rat striatal slice

1988 • 163 citations

The 5-HT3 receptor ligand, [3H]BRL 43694, binds to presynaptic sites in the nucleus tractus solitarius of the rat

1989 • 150 citations

Blockade of neuronal tryptamine receptors by metoclopramide

1978 • 148 citations

A 5-HT receptor in the central nervous system, positively coupled with adenylate cyclase, is antagonized by ICS 205 930

1988 • 137 citations

[3H]Quipazine labels 5-HT3 recognition sites in rat cortical membranes

1988 • 127 citations

Antiemetic properties of the 5HT3-receptor antagonist, gr38032f

1987 • 123 citations

Electrophysiological characterization of functionally distinct 5-hydroxytryptamine receptors on guinea-pig submucous plexus

1988 • 116 citations

Effect of the 5-HT3 receptor antagonist, GR38032F, on responses to injection of a neurokinin agonist into the ventral tegmental area of the rat brain

1987 • 113 citations

Neuroanatomical sites of action of 5‐HT₃ receptor agonist and antagonists for alteration of aversive behaviour in the mouse

1989 • 111 citations

Blockade of serotonin receptors on autonomic neurones by (−)-cocaine and some related compounds

1979 • 103 citations

Identification of serotonin 5-HT3 recognition sites by radioligand binding in NG108-15 neuroblastoma-glioma cells

1987 • 99 citations

5-HT3 receptor antagonists block morphine- and nicotine-induced place-preference conditioning

1988 • 98 citations

[3H]Quaternised ICS 205-930 labels 5-HT3 receptor binding sites in rat brain

1988 • 87 citations

A PHARMACOLOGICAL ANALYSIS OF THE MODE OF ACTION OF SEROTONIN (5‐HYDROXYTRYPTAMINE) UPON THE GUINEA‐PIG ILEUM

1953 • 78 citations

The dopamine response in mouse neuroblastoma cells is mediated by serotonin 5HT3 receptors

1986 • 56 citations

MEMBRANE POTENTIAL CHANGES INDUCED BY 5‐HYDROXYTRYPTAMINE IN THE RABBIT SUPERIOR CERVICAL GANGLION

1975 • 53 citations

Species variations in 5-HT3 recognition sites labeled by 3H-quipazine in the central nervous system

1988 • 38 citations

Influence of 5‐hydroxytryptamine uptake on the apparent 5‐hydroxytryptamine antagonist potency of metoclopramide in the rat isolated superior cervical ganglion

1987 • 32 citations

Prevention of physostigmine‐, DFP‐, and diazinon‐induced acute toxicity by monoethylcholine and N‐aminodeanol

1989 • 17 citations

Enhancement of leukotriene C₄ release from primate airway macrophages by cellular interactions

1989 • 16 citations