Adenosine Receptor Subtypes: Binding Studies

ADENOSINE REGULATES VIA TWO DIFFERENT TYPES OF RECEPTORS, THE ACCUMULATION OF CYCLIC AMP IN CULTURED BRAIN CELLS

1979 • 1,370 citations

Subclasses of external adenosine receptors.

1980 • 1,087 citations

Characterization of the A2 adenosine receptor labeled by [3H]NECA in rat striatal membranes.

1986 • 821 citations

Adenosine receptors in brain membranes: binding of N6-cyclohexyl[3H]adenosine and 1,3-diethyl-8-[3H]phenylxanthine.

1980 • 554 citations

Regulatory Function of Adenosine

1983 • 454 citations

Subclasses of adenosine receptors in the central nervous system: Interaction with caffeine and related methylxanthines

1983 • 437 citations

Adenosine and the concept of ‘retaliatory metabolites’

1984 • 422 citations

Binding of the A1-selective adenosine antagonist 8-cyclopentyl-1,3-dipropylxanthine to rat brain membranes

1987 • 376 citations

Characterization of adenosine receptors in rat brain by (?)[3H]N6-phenylisopropyladenosine

1980 • 296 citations

On the mechanism by which adenosine receptor activation inhibits the release of acetylcholine from motor nerve endings.

1984 • 214 citations

Regulation of adenosine formation by the heart.

1986 • 209 citations

Adenosine receptor activation in human fibroblasts: nucleoside agonists and antagonists

1980 • 198 citations

The character of the muscarinic receptors in different regions of the rat brain

1980 • 188 citations

Biochemical characterization of putative central purinergic receptors by using 2-chloro[3H]adenosine, a stable analog of adenosine.

1980 • 155 citations

Depression of Corticospinal Cells by Various Purines and Pyrimidines

1974 • 146 citations

Adenosine antagonism by purines, pteridines and benzopteridines in human fibroblasts

1981 • 137 citations

Adenosine receptors in fat cells. Identification by (-)-N6-[3H]phenylisopropyladenosine binding.

1981 • 118 citations

Adenosine receptors mediating cardiac depression

1982 • 115 citations

[3H]5?-N-ethylcarboxamide adenosine binds to both Ra and Ri adenosine receptors in rat striatum

1984 • 110 citations

Ligand selectivity of dog coronary adenosine receptor resembles that of adenylate cyclase stimulatory (Ra) receptors.

1983 • 110 citations

The dextro and levorotatory isomers of N-phenylisopropyladenosine: Stereospecific effects on cyclic AMP-formation and evoked synaptic responses in brain slices

1979 • 106 citations

Stereospecificity in some central and circulatory effects of phenylisopropyl-adenosine (PIA).

1975 • 99 citations

N6-Cycloalkyladenosines. Potent, A1-selective adenosine agonists

1985 • 98 citations

PD 115,199: An antagonist ligand for adenosine A2 receptors

1987 • 96 citations

[125I]Aminobenzyladenosine, a new radioligand with improved specific binding to adenosine receptors in heart.

1985 • 82 citations

Adenosine-sensitive adenylate cyclase in rat brain homogenates: kinetic characteristics, specificity, topographical, subcellular and cellular distribution.

1979 • 78 citations

Concentration dependency of the renal vascular and renin secretory responses to adenosine receptor agonists.

1985 • 75 citations

Nomenclature of adenosine receptors

1985 • 71 citations

1,3-Dipropyl-8-cyclopentylxanthine (DPCPX) inhibition of [3H]N-ethylcar☐amidoadenosine (NECA) binding allows the visualization of putative non-A1 adenosine receptors

1986 • 71 citations

Effects of adenosine derivatives on cAMP accumulation and lipolysis in rat adipocytes and on adenylate cyclase in adipocyte plasma membranes

1977 • 70 citations

5′‐N‐ETHYLCARBOXAMIDOADENOSINE: A POTENT INHIBITOR OF HUMAN PLATELET AGGREGATION

1981 • 69 citations

Regulation of breathing in the rat: Indications for a role of central adenosine mechanisms

1982 • 66 citations

Adenosine Receptors and Adenylate Cyclase Interactions

1983 • 57 citations

Electrophysiological responses to adenosine analogs in rat hippocampus and cerebellum: Evidence for mediation by adenosine receptors of the A1 subtype

1984 • 51 citations

Episodic release of renin from single isolated superfused rat afferent arterioles

1986 • 46 citations

Adenosine and Renal Function

1983 • 39 citations

Effects of several 5?-carboxamide derivatives of adenosine on adenosine receptors of human platelets and rat fat cells

1984 • 30 citations

Role of adenosine in cerebral metabolism and blood flow

1988 • 29 citations

[125I]Aminobenzyladenosine, a new radioligand with improved specific binding to adenosine receptors in heart.

1985 • 28 citations

Adenosine Analogues Stimulate Cyclic AMP‐Accumulation in Cultured Neuroblastoma and Glioma Cells

1984 • 28 citations

Adenosine-induced depression of synaptic transmission in the isolated olfactory cortex: receptor identification

1985 • 22 citations

Rat heart mitochondria release adenosine

1983 • 22 citations

Attempted antagonism of adenosine analogue induced depression of respiration

1984 • 17 citations

Coronary and cardiohemodynamic effects of 2-phenylamino-adenosine (CV-1808) in anesthetized dogs and cats.

1980 • 15 citations

N6-Functionalized congeners of adenosine with high potency at A2-adenosine receptors: Potential ligands for affinity chromatography

1986 • 7 citations