Stereochemistry of Dopamine Receptor Agonists

Brain dopamine receptors.

1980 • 1,878 citations

The Neurobiology of Dopamine

1980 • 496 citations

Dopamine receptor binding: Differentiation of agonist and antagonist states with 3H-dopamine and 3H-haloperidol

1975 • 390 citations

Dopamine receptors: Pharmacological and anatomical evidences indicate that two distinct dopamine receptor populations are present in rat striatum

1978 • 203 citations

Synthesis and pharmacology of some 2-aminotetralins. Dopamine receptor agonists

1975 • 134 citations

Cerebral dopamine agonist properties of some 2-aminotetralin derivatives after peripheral and intracerebral administration

1977 • 94 citations

Phenothiazine drugs: structure-activity relationships explained by a conformation that mimics dopamine.

1975 • 88 citations

Biochemical Actions of Neuroleptic Drugs: Focus on the Dopamine Receptor

1978 • 83 citations

Synthesis and dopaminergic activity of (+-)-, (+)-, and (-)-2-dipropylamino-5-hydroxy-1,2,3,4-tetrahydronaphthalene

1976 • 82 citations

Effects of some derivatives of 2-aminotetralin on dopamine-sensitive adenylate cyclase and on the binding of [3H]haloperidol to neuro-leptic receptors in the rat striatum

1978 • 50 citations

Evidence for essential thiol groups and disulfide bonds in agonist and antagonist binding to the dopamine receptor

1980 • 48 citations

Dopamine receptors in rat striatum and nucleus accumbens; conformational studies using rigid analogues of dopamine

1977 • 46 citations

Synthesis and biological activity of (6aS)-10,11-dihydroxyaporphine, the optical antipode of apomorphine

1973 • 46 citations

Mapping the dopamine receptor. 1. Features derived from modifications in ring E of the neuroleptic butaclamol

1979 • 44 citations

Neuroleptic agents of the benzocycloheptapyridoisoquinoline series. A hypothesis on their mode of interaction with the central dopamine receptor.

1975 • 40 citations

Monophenolic 2-(dipropylamino)indans and related compounds: central dopamine-receptor stimulating activity

1981 • 33 citations

Conformational analysis of dopamine by the INDO molecular orbital method

1977 • 32 citations

Neuroleptic receptors: Stereoselectivity for neuroleptic enantiomers

1979 • 30 citations

ENANTIOSELECTIVITY IN THE BINDING OF (+)- AND (−)-2-AMINO-6,7-DIHYDROXY-1,2,3,4-TETRAHYDRONAPHTHALENE AND RELATED AGONISTS TO DOPAMINE RECEPTORS

1979 • 28 citations

Congeners of the .beta. conformer of dopamine derived from cis- and trans-octahydrobenzo[f]quinoline and trans-octahydrobenzo[g]quinoline

1980 • 27 citations

Dopamine receptor binding for agonists and antagonists in thermal exposed membranes

1979 • 26 citations

The conformation of dopamine at its receptor: binding of monohydroxy-2-aminotetralin enantiomers and positional isomers.

1979 • 25 citations

Central Depressant Activity of Some Thiaxanthene Derivatives

1962 • 25 citations

Synthesis and stereospecific antipsychotic activity of (-)-1-cyclopropylmethyl-4-(3-trifluoromethylthio-5H-dibenzo[a,d]cyclohepten-5-ylidene)piperidine

1977 • 19 citations

Die absolute Konfiguration von (+)‐ und (–)‐2‐Amino‐tetralin sowie der vier isomeren 2‐Amino‐tetralole‐(1)

1969 • 18 citations

Antidepressants. Tetrabenazine-antagonizing activity in a series of 5H-dibenzo[cycloheptene-5-propylamines

1968 • 14 citations

ChemInform Abstract: THE CHEMISTRY OF DOPAMINE

1980 • 13 citations

2,3-Dihydroxy-9-amino-9,10-dihydrophenanthrene, a rigid congener of dopamine and isoapomorphine

1978 • 11 citations

ChemInform Abstract: MAPPING THE DOPAMINE RECEPTOR. 1. FEATURES DERIVED FROM MODIFICATIONS IN RING G E OF THE NEUROLEPTIC BUTACLAMOL

1979 • 8 citations

Neurotropic and psychotropic substances. XLII. 2-Hydroxy-9-(3-dimethylaminopropylidene)thioxanthenes and some related compounds

1970 • 8 citations

Butyrophenones and Diphenylbutylpiperidines

1974 • 7 citations

Butyrophenones and Diphenylbutylpiperidines

1980 • 7 citations

Evidence for, and localization of, a unitary dopamine receptor composed of cooperatively linked subunit binding sites in rat striatum.

1979 • 5 citations

ChemInform Abstract: CONGENERS OF THE β CONFORMER OF DOPAMINE DERIVED FROM CIS‐ AND TRANS‐OCTAHYDROBENZO(F)QUINOLINE AND TRANS‐OCTAHYDROBENZO(G)QUINOLINE

1980 • 1 citations