Synthesis and pharmacological evaluation of some amino-acid-containing cyproheptadine derivatives as dual antagonists of histamine H1- and leukotriene D4-receptors
Data up to Jan 2025
Total Citations Per Year
Abstract
References (18)
Histamine: an early messenger in inflammatory and immune reactions
1992 • 187 citations
Selective Type IV Phosphodiesterase Inhibitors as Antiasthmatic Agents. The Syntheses and Biological Activities of 3-(Cyclopentyloxy)-4-methoxybenzamides and Analogs
1994 • 113 citations
Complement research: biosynthesis, genetics, immunoregulatory role and clinical studies
1992 • 67 citations
Antihistamines in the treatment of asthma
1992 • 53 citations
Antagonists of slow reacting substance of anaphylaxis. Synthesis of a series of chromone-2-carboxylic acids
1977 • 49 citations
Structure-Activity Relationships in the Cyproheptadine Series
1965 • 47 citations
Interactions between leukotrienes and histamine in the anaphylactic contraction of guinea pig lung parenchyma.
1994 • 38 citations
Structure-activity relationships within a series of analogues of the histamine H1-antagonist terfenadine
1993 • 26 citations
(Piperidinylalkoxy)chromones: Novel Antihistamines with Additional Antagonistic Activity against Leukotriene D4
1995 • 25 citations
Synthesis of lactivicin analogues
1988 • 23 citations
Amphoteric Drugs. 3. Synthesis and Antiallergic Activity of 3-[(5,11-Dihydro[1]benzoxepino[4,3-b]pyridin-11-ylidene)piperidino]propionic Acid Derivatives and Related Compounds
1995 • 20 citations
Peptidoleukotriene Antagonists State of the Art
1992 • 18 citations
Dibenz[b,e]oxepin derivatives: novel antiallergic agents possessing thromboxane A2 and histamine H1 dual antagonizing activity. 1
1993 • 18 citations
QSAR and Molecular Modelling Studies on Histamine H1‐Receptor Antagonists
1992 • 17 citations
Discovery and preliminary pharmacology of Sch 37370, a dual antagonist of PAF and histamine
1991 • 13 citations
Antihistamines in the treatment of asthma
1994 • 11 citations
Optically active analogues of ebastine: Synthesis and effect of chirality on their antihistaminic and antimuscarinic activity
1994 • 5 citations
Histamine and Asthma
1990 • 3 citations