Classification of some GABA antagonists with regard to site of action and potency in slices of rat cuneate nucleus

Gamma-Aminobutyric Acid Binding to Receptor Sites in the Rat Central Nervous System

1974 • 589 citations

Antagonism between bicuculline and GABA in the cat brain

1971 • 363 citations

Characterization and ionic basis of GABA‐induced depolarizations recorded in vitro from cat primary afferent neurones.

1978 • 321 citations

Pentylenetetrazol and penicillin are selective antagonists of GABA-mediated post-synaptic inhibition in cultured mammalian neurones

1977 • 254 citations

DEPOLARIZING ACTIONS OF γ‐AMINOBUTYRIC ACID AND RELATED COMPOUNDS ON RAT SUPERIOR CERVICAL GANGLIA IN VITRO

1974 • 249 citations

Binding of [3H]alpha-dihydropicrotoxinin, a gamma-aminobutyric acid synaptic antagonist, to rat brain membranes.

1978 • 216 citations

GABA receptor binding with 3H (+) bicuculline–methiodide in rat CNS

1977 • 175 citations

Convulsive action of penicillin

1972 • 170 citations

GABA-picrotoxin interaction in the mammalian central nervous system

1969 • 164 citations

Evidence that bicuculline and picrotoxin act at separate sites to antagonize γ-aminobutyric acid in rat cuneate nucleus

1980 • 158 citations

CHARACTERIZATION OF THE BINDING OF [³H]MUSCIMOL, A POTENT γ‐AMINOBUTYRIC ACID AGONIST, TO RAT BRAIN SYNAPTOSOMAL MEMBRANES USING A FILTRATION ASSAY

1979 • 147 citations

The Receptors : a comprehensive treatise

1979 • 145 citations

Bicuculline Methochloride as a GABA Antagonist

1972 • 145 citations

Physiological identification of GABA as the inhibitory transmitter for mammalian cortical neurons in cell culture

1980 • 136 citations

The blockade of GABA mediated responses in the frog spinal cord by ammonium ions and furosemide.

1978 • 113 citations

MUSCIMOL UPTAKE, RELEASE AND BINDING IN RAT BRAIN SLICES

1978 • 102 citations

A comparative study of some convulsant substances as γ‐aminobutyric acid antagonists in the feline cerebral cortex

1973 • 101 citations

Penicillin and inhibition in the cat spinal cord

1972 • 99 citations

GAMMA‐AMINOBUTYRIC ACID BINDING IN MAMMALIAN BRAIN: RECEPTOR‐LIKE SPECIFICITY OF SODIUM‐INDEPENDENT SITES

1978 • 98 citations

Conductance increases produced by glycine and gamma‐aminobutyric acid in lamprey interneurones.

1978 • 98 citations

Synaptic Mechanism of Pentylenetetrazole: Selectivity for Chloride Conductance

1977 • 98 citations

PRESYNAPTIC ACTIONS OF β‐AMINOBUTYRIC ACID AND SOME ANTAGONISTS IN A SLICE PREPARATION OF CUNEATE NUCLEUS

1978 • 96 citations

Properties of gamma-aminobutyric acid receptor binding with (+)-[3H]bicuculline methiodide in rat cerebellum.

1978 • 93 citations

Chemical instability of the GABA antagonist bicuculline under physiological conditions

1975 • 89 citations

DISTINCTION BETWEEN THE EFFECTS OF BARBITURATES, BENZODIAZEPINES AND PHENYTOIN ON RESPONSES TO γ‐AMINOBUTYRIC ACID RECEPTOR ACTIVATION AND ANTAGONISM BY BICUCULLINE AND PICROTOXIN

1981 • 76 citations

Relationship between pentylenetetrazol-induced seizures and brain pentylenetetrazol levels in mice.

1980 • 72 citations

ANTAGONISM OF γ‐AMINOBUTYRIC ACID AND GLYCINE BY CONVULSANTS IN THE CUNEATE NUCLEUS OF CAT

1976 • 71 citations

A site for the potentiation of GABA-mediated responses by benzodiazepines

1980 • 70 citations

An analysis of [3H]gamma-aminobutyric acid (GABA) binding in the human brain

1979 • 66 citations

Convulsive Properties of d-Tubocurarine and Cortical Inhibition

1972 • 63 citations

Pentylenetetrazol: An antagonist of gaba at primary afferents of the isolated frog spinal cord

1976 • 55 citations

Antagonism by penicillin of γ-aminobutyric acid depolarizations at presynaptic sites in rat olfactory cortex and cuneate nucleus in vitro

1980 • 51 citations

The Pharmacon-Receptor-Effector Concept

1979 • 50 citations

Quantitative Aspects of Chemical Pharmacology

1979 • 43 citations

Bicuculline, benzyl penicillin, and inhibitory amino acids in the spinal cord of the cat

1977 • 41 citations

Substrate Specificity of [³H] Muscimol Binding to a Particulate Fraction of a Neuron‐enriched Culture of Embryonic Rat Brain

1980 • 28 citations

Antagonism of GABA by picrotoxin in the feline cerebral cortex

1972 • 26 citations

Quantitative aspects of chemical pharmacology

1980 • 23 citations

Some Observations on the Physical and Pharmacological Properties of Picrotoxin Solutions

1963 • 17 citations

A re-examination of the gaba-inhibitory action of bicuculline on lobster muscle

1981 • 17 citations

ANTAGONISM OF INHIBITORY AMINO ACID ACTION BY TUBOCURARINE

1974 • 16 citations

Neurotransmitters in Epilepsy

1988 • 14 citations

Chloride-dependent action of GABA on the infundibular-neurohypophysial compound action potential

1981 • 11 citations

Glycine and GABA induced conductance changes in lamprey reticulospinal neurons and their antagonism by strychnine, thebaine, bicuculline and picrotoxin

1979 • 10 citations