Back to search

Novel Agonists of 5HT2C Receptors. Synthesis and Biological Evaluation of Substituted 2-(Indol-1-yl)-1-methylethylamines and 2-(Indeno[1,2-b]pyrrol-1-yl)-1-methylethylamines. Improved Therapeutics for Obsessive Compulsive Disorder

Data up to Jan 2025

Published1997
Citations99
References20

Total Citations Per Year

Abstract

References (20)

LIGAND: A versatile computerized approach for characterization of ligand-binding systems

1980 • 8,534 citations

Interactions of selective serotonin reuptake inhibitors with the serotonin 5-HT2C receptor

1996 • 193 citations

Involvement of 5-HT1C-receptors in drug-induced penile erections in rats

1990 • 151 citations

Selective serotonin re-uptake inhibitors decrease schedule-induced polydipsia in rats: a potential model for obsessive compulsive disorder

1993 • 135 citations

Evidence for a role of 5-HT1C receptors in the antiserotonergic properties of some antidepressant drugs

1993 • 119 citations

Radiolabelling of the human 5-HT2A receptor with an agonist, a partial agonist and an antagonist: Effects on apparent agonist affinities

1996 • 80 citations

Methodology for the facile and regio-controlled synthesis of indoles

1983 • 66 citations

8-Hydroxy-2-(alkylamino)tetralins and related compounds as central 5-hydroxytryptamine receptor agonists

1984 • 59 citations

Rearrangements of chromanones and dihydrocoumarins by aluminium chloride

1954 • 48 citations

Synthesis and Pharmacological Activity of Fluorinated Tryptamine Derivatives

1963 • 37 citations

Synthesis and evaluation of a novel series of N,N-dimethylisotryptamines

1984 • 32 citations

BETA-PHENYLISOBUTYLMETHYL KETONE AND ITS DERIVATIVES. THE SYNTHESIS OF ALPHA- AND OF BETA-PHENYLISOVALERIANIC ACIDS

1929 • 22 citations

Steric effects in the synthesis of 1,7-dialkylindans

1986 • 17 citations

Acyltryptamines. II. Synthesis of Acyltryptamines, Indazoles, and Azepinoindoles from the Acylphenylhydrazones of 2,3-Piperidinedione1

1963 • 16 citations

Studies on Furan Compounds. I. Conversion of 2-Acetofuran to Hexen-2-dion-4,5-acetal-1 and Pyrocatechol

1948 • 15 citations

Preparation of Some Substituted β-Phenylisovaleric Acids

1948 • 11 citations

SYNTHESIS OF 1,1-DIMETHYLINDANE DERIVATIVES HAVING SYNTHETICALLY USEFUL SUBSTITUENTS AT THE 5- AND 6-POSITIONS

1978 • 5 citations

CONCERNING THE SYNTHESIS OF 4-METHOXYINDAN-1-ONE

1976 • 5 citations

ChemInform Abstract: Steric Effects in the Synthesis of 1,7‐Dialkylindans.

1986 • 2 citations

ChemInform Abstract: ZUR KENNTNIS EINIGER 2‐AMINOMETHYLIERTER KERNSUBSTITUIERTER INDANONE‐(1)

1973 • 1 citations

Cited By (0)

Loading...
Novel Agonists of 5HT2C Receptors. Synthesis and Biological Evaluation of Substituted… (1997) – Journal of Medicinal Chemistry | Metascience Observatory Explorer