Synthesis of [methoxy‐³H]‐ and [methoxy‐¹¹C]‐ labelled raclopride. Specific dopamine‐D₂ receptor ligands

Brain dopamine receptors.

1980 • 1,878 citations

Opposing roles for D-1 and D-2 dopamine receptors in efflux of cyclic AMP from rat neostriatum

1981 • 917 citations

Quantitative Analysis of D2 Dopamine Receptor Binding in the Living Human Brain by PET

1986 • 847 citations

Specific in vitro and in vivo binding of 3H-raclopride a potent substituted benzamide drug with high affinity for dopamine D-2 receptors in the rat brain

1985 • 503 citations

3H-spiroperidol labels dopamine receptors in pituitary and brain

1977 • 406 citations

Domperidone, a specific in vitro dopamine antagonist, devoid of in vivo central dopaminergic activity

1979 • 402 citations

Substituted benzamides as ligands for visualization of dopamine receptor binding in the human brain by positron emission tomography.

1985 • 304 citations

Remoxipride, a new potential antipsychotic compound with selective anti-dopaminergic actions in the rat brain

1984 • 213 citations

Spiperone: A ligand of choice for neuroleptic receptors

1978 • 178 citations

Preparation of 11C-labelled raclopride, a new potent dopamine receptor antagonist: Preliminary PET studies of cerebral dopamine receptors in the monkey

1985 • 141 citations

Some in vitro receptor binding properties of [3H]eticlopride, a novel substituted benzamide, selective for dopamine-D2 receptors in the rat brain

1985 • 127 citations

Substituted benzamide drugs as selective neuroleptic agents.

1981 • 122 citations

Effects of Remoxipride and some Related New Substituted Salicylamides on Rat Brain Receptors

1986 • 101 citations

Potential neuroleptic agents. 2,6-Dialkoxybenzamide derivatives with potent dopamine receptor blocking activities

1982 • 90 citations

Autoradiographic visualization of dopamine D-2 receptors in the monkey brain using the selective benzamide drug [3H]raclopride

1986 • 73 citations

Potential neuroleptic agents. 4. Chemistry, behavioral pharmacology, and inhibition of [3H]spiperone binding of 3,5-disubstituted N-[(1-ethyl-2-pyrrolidinyl)methyl]-6-methoxysalicylamides

1986 • 72 citations

Comparison of dopamine receptor sites labeled by [3H]-S-sulpiride and [3H]-spiperone in striatum.

1983 • 70 citations

Classification of drugs according to receptor binding profiles

1984 • 64 citations

Regional in vivo binding of the substituted benzamide [3H]eticlopride in the rat brain: Evidence for selective labelling of dopamine receptors

1986 • 64 citations

Contamination of serotonin-2 binding sites by an alpha-1 adrenergic component in assays with (3H) spiperone

1984 • 51 citations

Comparisons between the in Vitro Binding of Two Substituted Benzamides and Two Butyrophenones to Dopamine-D2 Receptors in the Rat Striatum

1986 • 32 citations

Preparation of tritium labelled benzamide dopamine‐D₂ lignads at high specific activity

1985 • 11 citations