Subclassification of α₁‐adrenoceptor recognition sites by urapidil derivatives and other selective antagonists

PROTEIN MEASUREMENT WITH THE FOLIN PHENOL REAGENT

1951 • 319,299 citations

THE ATTRACTIONS OF PROTEINS FOR SMALL MOLECULES AND IONS

1949 • 19,979 citations

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1973 • 12,522 citations

SOME QUANTITATIVE USES OF DRUG ANTAGONISTS

1959 • 3,948 citations

A practical computer-based approach to the analysis of radioligand binding experiments

1983 • 834 citations

α1Adrenoceptor subtypes linked to different mechanisms for increasing intracellular Ca2+ in smooth muscle

1987 • 482 citations

Characterization of alpha 1-adrenergic receptor subtypes in rat brain: a reevaluation of [3H]WB4104 and [3H]prazosin binding.

1986 • 456 citations

Evidence for more than one type of post-junctional α-Adrenoceptor

1982 • 399 citations

Comparison of alpha 1-adrenergic receptor subtypes distinguished by chlorethylclonidine and WB 4101.

1988 • 268 citations

Heterogeneity of alpha 1-adrenergic receptors revealed by chlorethylclonidine.

1987 • 267 citations

α1-Adrenoceptor subclassification in vascular smooth muscle

1986 • 215 citations

Biodata handling with microcomputers

1984 • 213 citations

5-Methyl-urapidil discriminates between subtypes of the α1-adrenoceptor

1988 • 208 citations

Differentiation of alpha 1-adrenergic receptors linked to phosphatidylinositol turnover and cyclic AMP accumulation in rat brain.

1987 • 104 citations

Urapidil and some analogues with hypotensive properties show high affinities for 5-hydroxytryptamine (5-HT) binding sites of the 5-HT1A subtype and for ?1-adrenoceptor binding sites

1987 • 78 citations

Central 5-HT1A Receptors and the Mechanism of the Central Hypotensive Effect of (+)8-OH-DPAT, DP-5-CT, R28935, and Urapidil

1988 • 62 citations

Identification of subtypes of [3H]prazosin-labelled receptor binding sites in rat brain

1985 • 52 citations

Effects of urapidil, clonidine, prazosin and propranolol on autonomic nerve activity, blood pressure and heart rate in anaesthetized rats and cats

1985 • 47 citations

Thyroid-dependent alterations of myocardial adrenoceptors and adrenoceptor-mediated responses in the rat

1985 • 45 citations

α-Adrenoceptor subclassification by classical and response-related methods: same question, different answers

1988 • 43 citations

Evidence for and against heterogeneity of alpha1-adrenoceptors

1986 • 43 citations

Cardiovascular effects and interaction with adrenoceptors of urapidil.

1985 • 41 citations

Adrenergic regulation of gluconeogenesis: possible involvement of two mechanisms of signal transduction in alpha 1-adrenergic action.

1985 • 39 citations

A comparison of the effects of doxazosin and alfuzosin with those of urapidil on preganglionic symphathetic nerve activity in anaesthetised cats

1986 • 36 citations

Hypotensive Effect of Urapidil: CNS Site and Relative Contribution

1987 • 31 citations

Are Drugs That Act Both on Serotonin Receptors and α1-Adrenoceptors More Potent Hypotensive Agents Than Those That Act Only on α1-Adrenoceptors?

1988 • 18 citations

α1-Adrenoceptors of rat myocardium: Comparison of agonist binding and positive inotropic response

1988 • 16 citations

Are Drugs That Act Both on Serotonin Receptors and α1-Adrenoceptors More Potent Hypotensive Agents Than Those That Act Only on α1-Adrenoceptors?

1988 • 12 citations

Limitations of Schild plots in a two-receptor system: alpha adrenoceptors of vascular smooth muscle.

1986 • 10 citations

Heterogeneity of alpha-1 Adrenergic Receptors

1987 • 7 citations