5-HT1-like receptor agonists enhance wakefulness

Quantitative autoradiographic mapping of serotonin receptors in the rat brain. I. Serotonin-1 receptors

1985 • 1,855 citations

Proposals for the classification and nomenclature of functional receptors for 5-hydroxytryptamine

1986 • 1,255 citations

The role of monoamines and acetylcholine-containing neurons in the regulation of the sleep-waking cycle

1972 • 1,091 citations

8-Hydroxy-2-(di-n-propylamino)-tetralin discriminates between subtypes of the 5-HT1 recognition site

1983 • 869 citations

The involvement of subtypes of the 5-HT1 receptor and of catecholaminergic systems in the behavioural response to 8-hydroxy-2-(di-n-Propylamino) tetralin in the rat

1984 • 678 citations

Two Distinct Central Serotonin Receptors with Different Physiological Functions

1981 • 640 citations

Receptor-binding properties in vitro and in vivo of ritanserin: A very potent and long acting serotonin-S2 antagonist.

1985 • 444 citations

Presynaptic 5-HT autoreceptors on serotonergic cell bodies and/or dendrites but not terminals are of the 5-HT1A subtype

1985 • 383 citations

Cardiovascular Effects of Serotonin Agonists and Antagonists

1990 • 234 citations

5-Hydroxytryptamine-2 antagonist increases human slow wave sleep

1986 • 231 citations

Serotonin release is modulated by presynaptic autoreceptors

1979 • 225 citations

Stereoselective blockade at [3H]5-HT binding sites and at the 5-HT autoreceptor by propranolol

1984 • 206 citations

The effect of para-chlorophenylalanine on the sleep of cats

1968 • 196 citations

Electrophysiologically-identified serotonin receptors in the rat CNS Effect of antidepressant treatment

1984 • 170 citations

5-HT: The Enigma Variations

1987 • 167 citations

Functional role of 5-HT2 receptors in the regulation of sleep and wakefulness in the rat

1989 • 139 citations

Serotonin autoreceptor in rat hippocampus: Pharmacological characterization as a subtype of the 5-HT1 receptor

1986 • 136 citations

Is pindolol a mixed agonist-antagonist at central serotonin (5-HT) receptors?

1986 • 131 citations

BMY 7378, a buspirone analog with high affinity, selectivity and low intrinsic activity at the 5-HT1A receptor in rat and guinea pig hippocampal membranes

1987 • 128 citations

Pharmacological analysis of the behavioural and thermoregulatory effects of the putative 5-HT1 receptor agonist, RU 24969, in the rat

1986 • 127 citations

5-HT2 receptors could be primarily involved in the regulation of slow-wabe sleep in the rat

1987 • 121 citations

The behavioural effects of RU 24969, a suggested 5-HT1 receptor agonist in rodents and the effect on the behaviour of treatment with antidepressants

1984 • 118 citations

The putative 5-HT1 receptor agonist, RU 24969, inhibits the efflux of 5-hydroxytryptamine from rat frontal cortex slices by stimulation of the 5-HT autoreceptor

1985 • 104 citations

Electrophysiological evidence that spiperone is an antagonist of 5-HT1A receptors in the dorsal raphe nucleus

1988 • 69 citations

Evidence that 8‐hydroxy‐2‐(n‐dipropylamino)tetralin (8‐OH‐DPAT) is a selective α₂‐adrenoceptor antagonist on guinea‐pig submucous neurones

1987 • 59 citations

Antagonistic properties of quipazine at presynaptic serotonin receptors and ?-adrenoceptors in rat brain cortex slices

1981 • 57 citations

MDL 72832: a potent and stereoselective ligand at central and peripheral 5-HT1A receptors

1988 • 54 citations

The distribution of serotonin binding sites in the hippocampal region of the rat brain. An autoradiographic study

1984 • 51 citations

Reserpine and sleep

1971 • 45 citations

Substituted piperazine and indole compounds increase extracellular serotonin in rat diencephalon as determined by in vivo microdialysis

1991 • 44 citations

Cyanopindolol is a highly potent and selective antagonist at the presynaptic serotonin autoreceptor in the rat brain cortex

1985 • 42 citations

Biochemical pharmacology of paradoxical sleep.

1983 • 42 citations

(−)-Propranolol and (±)-cyanopindolol are mixed agonists-antagonists at serotonin autoreceptors in the hippocampus of the rat brain

1987 • 41 citations

In vivo voltammetry in the suprachiasmatic nucleus of the rat: Effects of RU24969, methiothepin and ketanserin

1986 • 40 citations

Biochemical and electrophysiological evidence for an agonist action of CM 57493 at pre- and postsynaptic 5-hydroxytryptamine1A receptors in brain.

1989 • 40 citations

5-HT-CONTAINING NEURONS: UNIT ACTIVITY IN BEHAVING CATS

1973 • 40 citations

Disturbances of sleep and wakefulness associated with the use of antihypertensive agents

1987 • 38 citations

5HT1A agonist, 8-hydroxy-2-(DI-n-propylamino)tetralin (8-OH-DPAT), inhibits non-opioid analgesia in defeated mice: influence of route of administration

1989 • 37 citations

Species differences in the distribution of central 5-HT1 binding sites: a comparative autoradiographic study between rat and guinea pig

1991 • 36 citations

The effects of buspirone on sleep in the rat

1986 • 31 citations

Suppressant effects of selective 5-HT2 antagonists on rapid eye movement sleep in rats

1989 • 30 citations

The effect of alpha and beta adrenergic receptor blockers on sleep in the rat

1976 • 30 citations

Determination of the 5-HT receptor subtype involved in 8-OH-DPAT-induced hyperlocomotion: potential difficulties arising from inadequate pharmacological tools

1990 • 29 citations

N-(3-acetylaminophenyl)piperazine hydrochloride (BEA 1654), a putative 5-HT1 agonist, causes constriction of arteriovenous anastomoses and dilatation of arterioles

1985 • 26 citations

Influence of route of administration on potency of the selective 5HT-1A agonist, 8-hydroxy-2-(di-n-propylamino)tetralin, in rats.

1987 • 23 citations

The acute effects of reserpine on the sleep-wakefulness cycle in rabbits

1969 • 21 citations

Neurochemical and behavioural studies with RU-24969 in the rat

1988 • 19 citations

Effects of the?-adrenoceptor antagonists acebutolol and metoprolol on sleep pattern in normal subjects

1977 • 18 citations

Postsynaptic localization and up-regulation of serotonin 5-HT1D receptors in rat brain

1989 • 15 citations

Buspirone, 8-OH-DPAT and ipsapirone: effects on hippocampal cerebellar and sciatic fiber excitability

1988 • 11 citations

β-adrenoceptor blockade in rats enhances the ambulation induced by 5-HT1A receptor agonists

1989 • 11 citations

5-Hydroxyindoleacetic acid in cerebrospinal fluid: measurements in wakefulness, slow-wave and paradoxical sleep

1973 • 7 citations

Methiothepin enhances the potassium-evoked release of [3H]-noradrenaline in rat pineal gland

1987 • 6 citations

Effect of 10 days reserpine or apomorphine administration on sleep cycles in rats

1976 • 3 citations

Deleted Work

1955 • 0 citations