Differential interaction of antiestrogens with cytosol estrogen receptors

Estrogen-Receptor Interaction

1973 • 746 citations

Current Models of Steroid Hormone Action: A Critique

1976 • 707 citations

A MONOHYDROXYLATED METABOLITE OF TAMOXIFEN WITH POTENT ANTIOESTROGENIC ACTIVITY

1977 • 502 citations

A NEW DERIVATIVE OF TRIPHENYLETHYLENE: EFFECT ON IMPLANTATION AND MODE OF ACTION IN RATS

1967 • 456 citations

Uterine, cytoplasmic estrogen binding protein. Thermal stability and ligand dissociation rate. Assay of empty and filled sites by exchange

1973 • 288 citations

Oestrogen receptors and antagonism of steroid hormone action

1974 • 242 citations

Estrogen receptor · anti-estrogen complex: Atypical binding by uterine nuclei and effects on uterine growth

1973 • 195 citations

Estradiol-binding kinetics of the activated and nonactivated estrogen receptor.

1977 • 191 citations

Antiestrogen Action in the Uterus: Biological Ineffectiveness of Nuclear Bound Estradiol after Antiestrogen¹²³

1975 • 181 citations

Uterine bioassay of tamoxifen, trioxifene and a new estrogen antagonist (LY117018) in rats and mice

1980 • 137 citations

Studies on the mechanism of action of the nonsteroidal antioestrogen tamoxifen (I.C.I. 46,474) in the rat

1977 • 131 citations

Interaction of 17β-estradiol and its specific uterine receptor. Evidence for complex kinetic and equilibrium behavior

1971 • 130 citations

Different Nuclear Binding Sites for Antiestrogen and Estrogen Receptor Complexes¹,²

1977 • 117 citations

Interactions entre l'oestradiol et des sites récepteurs utérins

1970 • 90 citations

A Comparative Study of Antiestrogen Action: Temporal Patterns of Antagonism of Estrogen Stimulated Uterine Growth and Effects on Estrogen Receptor Levels¹²³

1977 • 86 citations

Estrogen Receptor Activation and the Dissociation Kinetics of Estradiol, Estriol, and Estrone*

1980 • 69 citations

High-affinity binding of the antiestrogen [3H]tamoxifen to the 8S estradiol receptor

1978 • 65 citations

Interaction of uterus cytosol receptor with estradiol equilibrium and kinetic studies

1971 • 60 citations

The Relevance of Interaction Kinetics in Determining Biological Response to Estrogens

1979 • 50 citations

The binding of tamoxifen to oestrogen receptor proteins under equilibrium and non-equilibrium conditions

1979 • 50 citations

Synthesis and antiestrogenic activity of [3,4-dihydro-2-(4-methoxyphenyl)-1-naphthalenyl][4-[2-(1-pyrrolidinyl)ethoxy]phenyl]methanone, methanesulfonic acid salt

1979 • 49 citations

The influence of synthetic anti-estrogens on the binding of tritiated estradiol-17β by cytosols of human uterus and human breast carcinoma

1973 • 47 citations

Absence of correlation between antiestrogenic activity and binding affinity for the estrogen receptor

1979 • 43 citations

Estradiol dependent decrease of binding inhibition by anti-estrogens (a possible test of receptor activation)

1977 • 34 citations

The effects of antioestrogens on the oestrogen receptor

1979 • 24 citations

Design of Anti-Hormones

1979 • 12 citations