Novel antioestrogens without partial agonist activity

Phenol red in tissue culture media is a weak estrogen: implications concerning the study of estrogen-responsive cells in culture.

1986 • 1,282 citations

Radioimmunoassay for Rat Luteinizing Hormone with Antiovine LH Serum and Ovine LH-131I

1968 • 878 citations

The pharmacology and clinical uses of tamoxifen

1984 • 873 citations

A NEW DERIVATIVE OF TRIPHENYLETHYLENE: EFFECT ON IMPLANTATION AND MODE OF ACTION IN RATS

1967 • 456 citations

Biochemical pharmacology of antiestrogen action.

1984 • 417 citations

Tamoxifen in advanced breast cancer

1978 • 343 citations

Activation, Transformation, and Subunit Structure of Steroid Hormone Receptors

1982 • 323 citations

CONTROLLED TRIAL OF TAMOXIFEN AS SINGLE ADJUVANT AGENT IN MANAGEMENT OF EARLY BREAST CANCER

1985 • 291 citations

Antagonism of estrogen action with a new benzothiophene derived antiestrogen

1983 • 244 citations

The agonistic-antagonistic properties of clomiphene: A review

1981 • 222 citations

Differential sensitivity of human breast cancer cell lines to the growth-inhibitory effects of tamoxifen.

1985 • 171 citations

THE PREVENTION OF BREAST CANCER

1986 • 143 citations

Uterine bioassay of tamoxifen, trioxifene and a new estrogen antagonist (LY117018) in rats and mice

1980 • 137 citations

Promoter Elements of Genes Coding for Proteins and Modulation of Transcription by Estrogens and Progesterone

1984 • 133 citations

DOUBLE-BLIND CONTROLLED TRIAL OF TAMOXIFEN THERAPY FOR MASTALGIA

1986 • 120 citations

New biospecific adsorbents for the purification of estradiol receptor.

1978 • 120 citations

Non-steroidal antioestrogens—Receptor binding and biological response in rat uterus, rat mammary carcinoma and human breast cancer cells

1984 • 110 citations

Pharmacology and clinical uses of inhibitors of hormone secretion and action

1987 • 91 citations

Non-Steroidal Antioestrogens

1983 • 72 citations

Abnormal Reproductive Development in Rats after Neonatally Administered Antiestrogen (Tamoxifen)

1979 • 61 citations

Estrogen-receptor binding and biologic activity of tamoxifen and its metabolites.

1980 • 59 citations

An evaluation of tamoxifen as a partial agonist by classical receptor theory — An explanation of the dual action of tamoxifen

1984 • 46 citations

PROLONGED OESTROGENIC AND MITOGENIC ACTIVITY OF TAMOXIFEN IN THE OVARIECTOMIZED MOUSE

1978 • 33 citations

Central action and a species comparison of the estrogenic effects of an antiestrogen on eating and body weight

1977 • 33 citations

The mechanism of action of oestrogens.

1985 • 32 citations

Receptor interconversion model of hormone action. I. ATP-mediated conversion of estrogen receptors from a high to lower affinity state and its relationship to antiestrogen action.

1986 • 24 citations

The estrogenic effects of clomiphene during the neonatal period in the rat

1983 • 17 citations

Tumor growth-stimulating and inhibiting effects of antiestrogens on the DMBA-induced mammary carcinoma of the ovariectomized, diethylstilbestrol-treated SD rat. A study on the mechanism of action of antiestrogens

1983 • 17 citations

Physicochemical characteristics of the interaction of the glucocorticoid antagonist RU38486 with glucocorticoid receptors in vitro, and the role of molybdate

1986 • 12 citations