5-HT-la and 5-HT-lb selectivity of two phenylpiperazine derivatives: Evidence for 5-HT-lb heterogeneity

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1973 • 12,522 citations

LIGAND: A versatile computerized approach for characterization of ligand-binding systems

1980 • 8,534 citations

Multiple serotonin receptors: differential binding of [3H]5-hydroxytryptamine, [3H]lysergic acid diethylamide and [3H]spiroperidol.

1979 • 1,321 citations

Psychopharmacology : a generation of progress

1978 • 1,168 citations

8-Hydroxy-2-(di-n-propylamino)-tetralin discriminates between subtypes of the 5-HT1 recognition site

1983 • 869 citations

Psychopharmacology: A generation of progress

1978 • 785 citations

Discrimination of Multiple [³H]5‐Hydroxytryptamine Binding Sites by the Neuroleptic Spiperone in Rat Brain

1981 • 629 citations

Validation and statistical analysis of a computer modeling method for quantitative analysis of radioligand binding data for mixtures of pharmacological receptor subtypes.

1982 • 573 citations

Characteristics of central 5-HT receptors and their adaptive changes following intracerebral 5,7-dihydroxytryptamine administration in the rat.

1978 • 336 citations

Stereoselective blockade at [3H]5-HT binding sites and at the 5-HT autoreceptor by propranolol

1984 • 206 citations

Comparison of the pharmacological characteristics of 5 HT1 and 5 HT2 binding sites with those of serotonin autoreceptors which modulate serotonin release

1982 • 200 citations

Disposition and pharmacological effects of m-Chlorophenylpiperazine in rats

1981 • 127 citations

Molecular Pharmacology of Neurotransmitter Receptors

1984 • 122 citations

Selective Anti-Aggressive Properties of DU 27725: Ethological Analyses of Intermale and Territorial Aggression in the Male Rat

1981 • 107 citations

[³H]5‐Hydroxytryptamine Binding Sites: Species and Tissue Variation

1984 • 105 citations

Serotonin-induced contraction of canine basilar artery: mediation by 5-HT1 receptors

1983 • 76 citations

Plasma concentrations of trazodone and 1-(3-chlorophenyl)piperazine in man after a single oral dose of trazodone

1982 • 69 citations

Structural relationships in the inhibition of [3H]serotonin binding to rat brain membranes in vitro by 1-phenyl-piperazines

1980 • 54 citations

Antagonism of vascular serotonin receptors by m-chlorophenylpiperazine and m-trifluoromethylphenylpiperazine

1983 • 50 citations

Dual Effects of Ascorbate on Serotonin and Spiperone Binding in Rat Cortical Membranes

1983 • 44 citations

Anti-aggressive effect of a new phenylpiperazine compound (DU27716) on hypothalamically induced behavioural activities

1982 • 44 citations

Differential effect of cholesterol on two types of 5-hydroxytryptamine binding sites

1983 • 27 citations

Molecular pharmacology of neurotransmitter receptors

1983 • 22 citations

Photoaffinity labeling of serotonin-binding proteins

1979 • 18 citations