An Enantioselective Ketene−Imine Cycloaddition Method for Synthesis of Substituted Ring-Fused 2-Pyridinones

Comprehensive Heterocyclic Chemistry

1984 • 2,966 citations

Free Radical Damage and its Control

1994 • 297 citations

Total synthesis of elfamycins: aurodox and efrotomycin. 1. Strategy and construction of key intermediates

1985 • 142 citations

Synthesis of isotopically labelled 3-amino-2-phenylpropionic acid and its role as a precursor in the biosynthesis of tenellin and tropic acid

1991 • 98 citations

N- vs. O-alkylation in the mitsunobu reaction of 2-pyridone

1994 • 87 citations

Controlling Polymerization of β-Amyloid and Prion-derived Peptides with Synthetic Small Molecule Ligands

2000 • 69 citations

Titanium(IV)-Mediated Tandem Deprotection−Cyclodehydration of Protected Cysteine N-Amides: Biomimetic Syntheses of Thiazoline- and Thiazole-Containing Heterocycles

2000 • 67 citations

Preparation of highly substituted 2-pyridones by reaction of vinyl isocyanates and enamines

1989 • 66 citations

Synthesis of .alpha.-Pyridone-Based Azaheteroaromatics by Intramolecular Vinylketene Cyclizations onto the C:N Bond of Nitrogen Heteroaromatics

1994 • 64 citations

Ueber einige Ammoniumverbindungen

1892 • 55 citations

Therapeutic approaches to Alzheimer’s disease

2000 • 54 citations

Isolation of A58365A and A58365B, angiotensin converting enzyme inhibitors produced by Streptomyces chromofuscus.

1985 • 48 citations

Substituted 2-pyrones, 2-pyridones, and other congeners of elasnin as potential agents for the treatment of chronic obstructive lung diseases

1985 • 48 citations

Structure elucidation of A58365A and A58365B, angiotensin converting enzyme inhibitors produced by Streptomyces chromofuscus.

1988 • 48 citations

Mimicry of Peptide Backbone Geometry and Heteroatomic Side-Chain Functionality: Synthesis of Enantiopure Indolizidin-2-one Amino Acids Possessing Alcohol, Acid, and Azide Functional Groups

2001 • 47 citations

Synthesis of Six-membered Rings

1984 • 46 citations

Stereoselective Synthesis of Optically Active β-Lactams, Potential Inhibitors of Pilus Assembly in Pathogenic Bacteria

2000 • 43 citations

A photochemical [4+4] method for the construction of annulated eight-membered rings

1991 • 42 citations

Reaction ofa-KetoketeneS,N-Acetals with Cyanoacetamide: A New General Method for Substituted and Fused 4-(N-Alkylamino-,N-Arylamino-, orN-Morpholino)-3-cyano-2(1H)-pyridones

1982 • 38 citations

Oxazolines XXIV: Chiral Oxazolines and Thiazolines from L-Serine and L-Cysteine. Their Potential Use in Asymmetric Synthesis

1976 • 32 citations

Reformatskii reaction on .alpha.-oxo ketene dithioacetals: synthesis of substituted and fused ethyl 2-hydroxy-6-(methylthio)benzoates, 6-(methylthio)pyran-2-ones, and 6-(methylthio)-2(1H)pyridone derivatives

1990 • 31 citations

A new antibiotic produced by a strain of aspergillus flavipes

1968 • 30 citations

Methods for the detection and quantitation of angiotensin converting enzyme inhibitors in fermentation broths.

1985 • 30 citations

Reactions de michael sur des amides α,β insatures activees par le systeme CsF/Si(OCH3)4

1986 • 29 citations

Intramolecular [4 + 4] photocycloaddition of 2-pyridones tethered by a three-carbon chain: studies on the formation of cycloadducts and control of stereogenesis. 3

1994 • 27 citations

Stable carbocations. 184. 2,4-Dehydro-5-homoadamantyl cations

1976 • 19 citations

A Facile Synthesis of Substituted 4-Hydroxy-2-pyridones

1991 • 19 citations

Ester-Imine Condensation Mediated by Potassiumtert-Butoxide: Synthesis of β-Lactams and 3,4-Dihydropyridin-2-ones

1994 • 15 citations

Investigations on Pantothenic Acid and Its Related Compounds. III. Chemical Studies. (2). Synthesis of Di-D-pantothenoyl-L-cystine

1967 • 10 citations

A novel [3,3]-rearrangement of 1,2-dihydro-N-(arylamino)pyridines. Formation of unusual fused indolines

1986 • 7 citations

Rearrangement of 2-(haloalkoxy)pyridines to N-haloalkyl-2(1H)-pyridones

1993 • 6 citations

Synthesis and nuclear magnetic resonance study of 2-thiazolines

1984 • 6 citations

Structure of a new 1,4-diphenyl-3H-2-benzopyran-3-one derivative

1984 • 2 citations