[125I]Iodoproxyfan and Related Compounds: A Reversible Radioligand and Novel Classes of Antagonists with High Affinity and Selectivity for the Histamine H3 Receptor
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References (20)
Gravitational-wave bursts with memory and experimental prospects
1987 • 307 citations
Histamine H3 receptor-mediated inhibition of serotonin release in the rat brain cortex
1988 • 304 citations
Histamine H3 receptors modulate the release of [3H]‐acetylcholine from slices of rat entorhinal cortex: evidence for the possible existence of H3 receptor subtypes
1992 • 256 citations
Involvement of histamine in the control of the waking state
1993 • 164 citations
Three loci related to the src oncogene and tyrosine-specific protein kinase activity in Drosophila
1983 • 124 citations
Characterization and tissue distribution of H3 histamine receptors in guinea pigs by Nα-methylhistamine
1990 • 93 citations
Effect of thioperamide, a histamine H3 receptor antagonist, on electrically induced convulsions in mice
1993 • 84 citations
Synthesis, configuration, and calcium modulatory properties of enantiomerically pure 5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylates
1992 • 76 citations
Trichloromethyl chloroformate. Reaction with amines, amino acids, and amino alcohols
1976 • 71 citations
Characterization of the binding of the first selective radiolabeled histamine H3‐receptor antagonist, [125I]‐iodophenpropit, to rat brain
1994 • 63 citations
Iodoaminopotentidine and related compounds: a new class of ligands with high affinity and selectivity for the histamine H2 receptor
1992 • 53 citations
Novel histamine H3 receptor antagonists: affinities in an H3 receptor binding assay and potencies in two functional H3 receptor models
1994 • 49 citations
The first radiolabeled histamine H3 receptor antagonist, [125I]iodophenpropit: Saturable and reversible binding to rat cortex membranes
1992 • 48 citations
Responses of Anterior Pituitary Hormones and Hypothalamic Histamine to Blockade of Histamine Synthesis and to Selective Activation or Inactivation of Presynaptic Histamine H<sub>3</sub> Receptors in Stressed Rats
1993 • 30 citations
Unsymmetrically substituted guanidines as potent histamine H3-receptor antagonists
1994 • 21 citations
Acylated and alkylated histamine derivatives as new histamine H3-receptor antagonists
1994 • 19 citations
A convenient preparation of 3‐(1H‐imidazol‐4‐yl)propanol
1975 • 17 citations
An electron spin resonance study of the radical anion of 7,8-dimethylene-1,3,5-cyclooctatriene
1976 • 15 citations
New potent histamine H3-receptor antagonists of the amide type
1995 • 10 citations
Effects of iodoproxyfan, a potent and selective histamine H3 receptor antagonist, onα 2 and 5-HT3 receptors
1995 • 8 citations