Adenosine receptors and their ligands

Actions of caffeine in the brain with special reference to factors that contribute to its widespread use.

1999 • 2,431 citations

Nomenclature and classification of purinoceptors.

1994 • 1,569 citations

The physiological activity of adenine compounds with especial reference to their action upon the mammalian heart1

1929 • 1,470 citations

ADENOSINE REGULATES VIA TWO DIFFERENT TYPES OF RECEPTORS, THE ACCUMULATION OF CYCLIC AMP IN CULTURED BRAIN CELLS

1979 • 1,370 citations

Subclasses of external adenosine receptors.

1980 • 1,087 citations

Aggressiveness, hypoalgesia and high blood pressure in mice lacking the adenosine A2a receptor

1997 • 906 citations

The effect of adenosine and adenine nucleotides on the cyclic adenosine 3', 5'-phosphate content of guinea pig cerebral cortex slices.

1970 • 860 citations

Adenosine receptors: targets for future drugs

1982 • 681 citations

Molecular cloning and characterization of an adenosine receptor: the A3 adenosine receptor.

1992 • 649 citations

Molecular cloning and characterization of the human A3 adenosine receptor.

1993 • 421 citations

Cloned adenosine A3 receptors: Pharmacological properties, species differences and receptor functions

1994 • 395 citations

Adenosine inhibits the accumulation of cyclic AMP in cultured brain cells

1978 • 251 citations

[(3)H]MRE 3008F20: a novel antagonist radioligand for the pharmacological and biochemical characterization of human A(3) adenosine receptors.

2000 • 149 citations

Functional characterization of the A2b adenosine receptor in NIH 3T3 fibroblasts

1994 • 140 citations

2-Chloro-N6-[3H]cyclopentyladenosine ([3HCCPA) ?a high affinity agonist radioligand for A1 adenosine receptors

1989 • 131 citations

Water-Soluble Phosphate Prodrugs of 1-Propargyl-8-styrylxanthine Derivatives, A_2A-Selective Adenosine Receptor Antagonists

2000 • 119 citations

Biochemical characterization of the triazoloquinazoline, CGS 15943, a novel, non-xanthine adenosine antagonist.

1987 • 112 citations

Metabolic flux rates of adenosine in the heart

2000 • 111 citations

Search for New Purine- and Ribose-Modified Adenosine Analogs as Selective Agonists and Antagonists at Adenosine Receptors

1995 • 94 citations

125I-4-(2-[7-amino-2-[2-furyl][1,2,4]triazolo[2,3-a][1,3,5] triazin-5-yl-amino]ethyl)phenol, a high affinity antagonist radioligand selective for the A2a adenosine receptor.

1995 • 88 citations

New substituted 9-alkylpurines as adenosine receptor ligands

1998 • 78 citations

Use of the triazolotriazine [3H]ZM 241385 as a radioligand at recombinant human A2B adenosine receptors.

1999 • 70 citations

Adenosine A1 receptors in mammalian brain: Species differences in their interactions with agonists and antagonists

1986 • 66 citations

Characterization of human A_2A adenosine receptors with the antagonist radioligand [³H]‐SCH 58261

1997 • 63 citations

Comparison of A1 adenosine receptors in brain from different species by radioligand binding and photoaffinity labelling

1991 • 60 citations

Species differences in high‐affinity adenosine A₂ binding sites in striatal membranes from mammalian brain

1988 • 60 citations

[3H]-MRE 3008-F20: a novel antagonist radioligand for the pharmacological and biochemical characterization of human A3 adenosine receptors.

2000 • 59 citations