Enhancement of GABA binding by the benzodiazepine partial agonist CGS9896

GABAergic modulation of benzodiazepine binding site sensitivity

1978 • 726 citations

Molecular Mechanisms in the Receptor Action of Benzodiazepines

1979 • 579 citations

Benzodiazepine recognition site ligands: biochemistry and pharmacology.

1983 • 244 citations

Effects of drugs on γ-aminobutyric acid receptors, uptake, release and synthesis in vitro

1978 • 205 citations

Novel non-benzodiazepine anxiolytics

1983 • 109 citations

Enhancement of benzodiazepine and GABA binding by the novel anxiolytic, tracazolate

1982 • 93 citations

CGS 9896: A nonbenzodiazepine, nonsedating potential anxiolytic

1984 • 68 citations

Photoaffinity labeling of benzodiazepine receptors causes altered agonist-antagonist interactions

1983 • 41 citations

Modulation by calcium of gamma-aminobutyric acid (GABA) binding to GABAA and GABAB recognition sites in rat brain. Involvement of different mechanisms.

1984 • 39 citations

1,4-Benzodiazepines and Gamma-Aminobutyric Acid: Pharmacological and Biochemical Correlates

1979 • 38 citations

Photoaffinity labelling of the benzodiazepine receptor cannot be used to predict ligand efficacy

1983 • 30 citations

In vivo determination of efficacy of pyrazoloquinolinones at the benzodiazepine receptor

1984 • 24 citations

Modulation of GABA Receptor Binding by Ca⁺²

1983 • 23 citations

Distinction of benzodiazepine receptor agonists and inverse agonists by binding studies in vitro.

1983 • 22 citations

Modification of pyrazoloquinolinone affinity by GABA predicts efficacy at the benzodiazepine receptor

1984 • 16 citations

Benzodiazepines stimulate muscimol receptor binding in an Ro 15-1788 reversible manner

1983 • 11 citations