Antagonism of GABA_B‐receptor‐mediated responses in the guinea‐pig isolated ileum and vas deferens by phosphono‐analogues of GABA

3H-baclofen and 3H-GABA bind to bicuculline-insensitive GABAB sites in rat brain

1981 • 1,044 citations

GABAA and GABAB receptor site distribution in the rat central nervous system

1987 • 865 citations

KINETIC PARAMETERS OF NARCOTIC AGONISTS AND ANTAGONISTS, WITH PARTICULAR REFERENCE TO N‐ALLYLNOROXYMORPHONE (NALOXONE)

1968 • 392 citations

Bicuculline-insensitive gaba receptors on peripheral autonomic nerve terminals

1981 • 376 citations

Pre- and postsynaptic GABAB receptors in the hippocampus have different pharmacological properties

1988 • 368 citations

Phaclofen: a peripheral and central baclofen antagonist

1987 • 349 citations

The pharmacology of amino acids related to gamma-aminobutyric acid.

1965 • 333 citations

2-Hydroxy-saclofen: an improved antagonist at central and peripheral GABAB receptors

1988 • 202 citations

GABAergic mechanisms in the mammalian periphery

1987 • 197 citations

PRESYNAPTIC γ‐AMINOBUTYRIC ACID RECEPTORS IN THE RAT ANOCOCCYGEUS MUSCLE AND THEIR ANTAGONISM BY 5‐AMINOVALERIC ACID

1982 • 122 citations

Baclofen antagonism by 2-hydroxy-saclofen in the cat spinal cord

1988 • 78 citations

Comparison of antagonism by phaclofen of baclofen induced hyperpolarizations and synaptically mediated late hyperpolarizing potentials recorded intracellularly from rat dorsolateral septal neurons

1988 • 66 citations

Evidence for pharmacologically distinct subsets of GABAB receptors

1988 • 63 citations

Synthesis and pharmacological evaluation of .gamma.-aminobutyric acid analogs. New ligand for GABAB sites

1987 • 54 citations

Homotaurine: a GABA_B antagonist in guinea‐pig ileum

1983 • 52 citations

GABAA and GABAB receptors in locus coeruleus: effects of blockers

1988 • 49 citations

Glutamate transmitter in the central nervous system

1982 • 45 citations

The Synthesis of Phosphonobaclofen, an Antagonist of Baclofen

1987 • 32 citations

GABAB-receptor-mediated actions of baclofen in rat isolated neocortical slice preparations: antagonism by phosphono-analogues of GABA

1989 • 29 citations

Interactions between GABA and 5-hydroxytryptamine in the guinea-pig ileum

1983 • 27 citations

Phaclofen antagonizes baclofen-induced suppression of visually evoked responses in the cat's striate cortex

1988 • 27 citations

Benzofuran analogues of baclofen: a new class of central and peripheral GABAB-receptor antagonists

1989 • 26 citations

Phaclofen antagonizes GABA at autoreceptors regulating release in rat cerebral cortex

1988 • 26 citations

Differing actions of β-phenyl-GABA and baclofen in the guinea pig isolated ileum

1987 • 20 citations

Neuroactive properties of phosphonic amino acids

1979 • 20 citations

Baclofen antagonism by 4-amino-3-(5-methoxybenzo[b]furan-2-yl) butanoic acid in the cat spinal cord

1989 • 18 citations

Phosphorus analogs of .gamma.-aminobutyric acid, a new class of anticonvulsants

1984 • 16 citations

GABA‐RELATED ACTIVITIES OF AMINO PHOSPHONIC ACIDS ON GUINEA‐PIG ILEUM LONGITUDINAL MUSCLE

1986 • 13 citations