Session 2: Histamine Receptors: An Overview

Definition and Antagonism of Histamine H2-receptors

1972 • 2,284 citations

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

1983 • 1,548 citations

Highly potent and selective ligands for histamine H3-receptors

1987 • 890 citations

The physiological action of β‐iminazolylethylamine

1910 • 867 citations

RECEPTORS MEDIATING SOME ACTIONS OF HISTAMINE

1966 • 762 citations

pA, A NEW SCALE FOR THE MEASUREMENT OF DRUG ANTAGONISM

1947 • 759 citations

Pharmacology of Histamine Receptors

1982 • 375 citations

Metiamide — An orally active histamine H2-receptor antagonist

1973 • 259 citations

Association of long lasting unsurmountable histamine H2 blockade and gastric carcinoid tumours in the rat.

1985 • 242 citations

Dimaprit-[S-[3-(N,N-dimethylamino)propyl]isothiourea] —A highly specific histamine H2-receptor agonist. Part 1. Pharmacology

1977 • 240 citations

Histamine shock

1919 • 226 citations

Impromidine (SK&F 92676) is a very potent and specific agonist for histamine H2 receptors

1978 • 220 citations

An analysis of the responses of the isolated stomach to electrical stimulation and to drugs

1963 • 218 citations

Characterization and development of cimetidine as a histamine H2-receptor antagonist

1978 • 203 citations

The action of histamine and 5-hydroxytryptamine on isolated mammalian atria.

1960 • 177 citations

β-imidazolyläthylamin und die Organextrakte

1920 • 159 citations

Chemistry and Structure—Activity Relationships of Drugs Acting at Histamine Receptors

1982 • 133 citations

Further observations on the action of β‐iminazolylethylamine

1911 • 126 citations

PHARMACOLOGY OF ANTIHISTAMINE COMPOUNDS

1947 • 120 citations

Histamine H₃‐receptors inhibit cholinergic neurotransmission in guinea‐pig airways

1989 • 110 citations

Observations on Reactive Hyperaemia as Related to Histamine, on Drugs Antagonizing Vasodilatation Induced by Histamine and on Vasodilator Properties of Adenosinetri phosphate

1948 • 89 citations

H1+H2-receptor antagonists for premedication in anaesthesia and surgery: A critical view based on randomized clinical trials with haemaccel and various antiallergic drugs

1980 • 82 citations

HISTAMINE RECEPTORS IN PERIPHERAL VASCULAR BEDS IN THE CAT

1975 • 74 citations

Ranitidine (AH 19065): a new potent, selective histamine H2-receptor antagonist [proceedings].

1979 • 73 citations

THE ANTIHISTAMINE SUBSTANCE 2786 R.P.

1946 • 55 citations

The anti-histamine properties of benadryl, beta-di-methylaminoethyl benzhydryl ether hydrochloride.

1946 • 45 citations

Atypical (relaxant) response to histamine in cat bronchus

1977 • 34 citations

Potential histamine H2-receptor antagonists. 2. N.alpha.-Guanylhistamine

1975 • 33 citations

EVIDENCE FOR BOTH HISTAMINE H₁‐ AND H₂‐RECEPTORS IN THE GASTRIC VASCULATURE OF THE CAT

1980 • 33 citations

3-[4(5)-Imidazolyl] propylguanidine (SK&F 91486) — a partial agonist at histamine H2-receptors

1975 • 31 citations

H₁‐ AND H₂‐RECEPTORS IN THE SMOOTH MUSCLE OF THE RUMINANT STOMACH

1978 • 21 citations

The effects of prenylamine on single ventricular myocytes of guinea‐pig

1988 • 16 citations

Comparison of antisecretory potency and duration of action of the H2-receptor antagonists AH 22216, cimetidine, ranitidine and SK & F 93479 in the dog

1983 • 14 citations

Topics in gastroenterology 15

1988 • 2 citations