Back to search

Comparative pharmacological studies of melatonin receptors: mt1, mt2 and mt3/qr2. tissue distribution of mt3/qr2 11Abbreviations: MCA-NAT, methoxy-carbonylamino-N-acetyltrypta- mine, 2-[125I]-I-MCA-NAT, 2-[125I]-iodomethoxy-carbonylamino-N-acetyltryptamine; 2-IbMT, 2-iodo-N-butanoyl-5-methoxytryptamine; 4-P-PDOT, 4-phenyl-2-propionamido-tetraline; DH97, N-pentanoyl-2-benzyltryptamine; S20760, 5-methoxy-N-cyclopropanoyl-tryptamine; S24635, N-[2-(5-carbamoylbenzofuran-3-yl)ethyl]-acetamide; …

Data up to Jan 2025

Published2001
Citations186
References39

Total Citations Per Year

Abstract

References (39)

PROTEIN MEASUREMENT WITH THE FOLIN PHENOL REAGENT

1951 • 319,299 citations

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1973 • 12,522 citations

Cloning and characterization of a mammalian melatonin receptor that mediates reproductive and circadian responses

1994 • 1,099 citations

Molecular characterization of a second melatonin receptor expressed in human retina and brain: the Mel1b melatonin receptor.

1995 • 878 citations

Melatonin receptors: Localization, molecular pharmacology and physiological significance

1994 • 615 citations

Identification of the Melatonin-binding SiteMT 3 as the Quinone Reductase 2

2000 • 589 citations

Free-Running Activity Rhythms in the Rat: Entrainment by Melatonin

1983 • 552 citations

The immunoneuroendocrine role of melatonin

1993 • 493 citations

Expression cloning of a high-affinity melatonin receptor from Xenopus dermal melanophores.

1994 • 434 citations

Melatonin receptors: Are there multiple subtypes?

1995 • 410 citations

Selective MT 2 melatonin receptor antagonists block melatonin‐mediated phase advances of circadian rhythms

1998 • 357 citations

Melatonin receptor antagonists that differentiate between the human Mel1a and Mel1b recombinant subtypes are used to assess the pharmacological profile of the rabbit retina ML1 presynaptic heteroreceptor

1997 • 320 citations

Dual Signaling of Human Mel1a Melatonin Receptors via Gi2, Gi3, and Gq/11 Proteins

1999 • 258 citations

4-(3-Cyclopentyloxy-4-methoxyphenyl)-2-pyrrolidone (ZK 62711): a potent inhibitor of adenosine cyclic 3',5'-monophosphate phosphodiesterases in homogenates and tissue slices from rat brain.

1976 • 222 citations

Characterization of high‐affinity melatonin binding sites in purified cell nuclei of rat liver

1994 • 190 citations

Iodinated melatonin: Preparation and characterization of the molecular structure by mass and 1H NMR spectroscopy

1984 • 175 citations

Differential signaling of human Mel1a and Mel1b melatonin receptors through the cyclic guanosine 3′-5′-monophosphate pathway

1999 • 160 citations

Prazosin Update A Review of its Pharmacological Properties and Therapeutic Use in Hypertension and Congestive Heart Failure

1983 • 154 citations

Synthesis and Structure-Activity Relationships of Novel Naphthalenic and Bioisosteric Related Amidic Derivatives as Melatonin Receptor Ligands

1994 • 148 citations

Melatonin madness

1995 • 146 citations

2-[125I]Iodomelatonin Binding Sites in Hamster Brain Membranes: Pharmacological Characteristics and Regional Distribution*

1988 • 134 citations

Unexpected genetic and structural relationships of a long-forgotten flavoenzyme to NAD(P)H:quinone reductase (DT-diaphorase)

1997 • 121 citations

Human NAD(P)H:quinone oxidoreductase2. Gene structure, activity, and tissue-specific expression.

1994 • 117 citations

2-[125I]Iodo-5-methoxycarbonylamino-N-acetyltryptamine: a selective radioligand for the characterization of melatonin ML2 binding sites

1996 • 111 citations

Melatonin receptor density is regulated in rat pars tuberalis and suprachiasmatic nuclei by melatonin itself

1993 • 99 citations

Therapeutic potential of analogues of amiloride: inhibition of the regulation of intracellular pH as a possible mechanism of tumour selective therapy

1993 • 80 citations

Pharmacological characterization of melatonin binding sites in Syrian hamster hypothalamus

1990 • 78 citations

Characterization of 2-[125I]iodomelatonin binding sites in Syrian hamster peripheral organs.

1999 • 78 citations

Melatonin, Its Receptors, and Relationships with Biological Rhythm Disorders

1997 • 77 citations

Characterization of central melatonin receptors using 125I‐melatonin

1986 • 76 citations

Melatonin Receptors in Peripheral Tissues: A New Area of Melatonin Research

1993 • 74 citations

Specific binding of melatonin by purified cell nuclei from spleen and thymus of the rat

1998 • 66 citations

Comparison of the structure-activity relationships of melatonin receptor agonists and antagonists: lengthening the N-acyl side-chain has differing effects on potency on Xenopus melanophores

1998 • 50 citations

GR196429: a nonindolic agonist at high-affinity melatonin receptors.

1998 • 42 citations

Mouse NRH:quinone oxidoreductase (NQO2): cloning of cDNA and gene- and tissue-specific expression

2000 • 34 citations

Characterization of a melatonin binding site in Siberian hamster brown adipose tissue

1997 • 31 citations

Are nuclear receptors involved in pituitary responsiveness to melatonin?

1996 • 25 citations

[3H](+)S 14297: A novel, selective radioligand at cloned human dopamine D3 receptors

1995 • 10 citations

[Melatonin and regulation of the cardiovascular system].

1999 • 10 citations

Cited By (0)

Loading...
Comparative pharmacological studies of melatonin receptors: mt1, mt2 and mt3/qr2. tissue… (2001) – Biochemical Pharmacology | Metascience Observatory Explorer