Characterization of histamine‐H₃ receptors controlling non‐adrenergic non‐cholinergic contractions of the guinea‐pig isolated ileum

SOME QUANTITATIVE USES OF DRUG ANTAGONISTS

1959 • 3,948 citations

Simultaneous analysis of families of sigmoidal curves: application to bioassay, radioligand assay, and physiological dose-response curves.

1978 • 2,400 citations

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

1983 • 1,548 citations

Highly potent and selective ligands for histamine H3-receptors

1987 • 890 citations

RECEPTORS MEDIATING SOME ACTIONS OF HISTAMINE

1966 • 762 citations

Histamine H3 receptor-mediated inhibition of serotonin release in the rat brain cortex

1988 • 304 citations

STIMULANT ACTIONS OF VOLATILE ANAESTHETICS ON SMOOTH MUSCLE

1964 • 261 citations

Inhibition of noradrenaline release in the rat brain cortex via presynaptic H3 receptors

1989 • 245 citations

Competitive antagonists discriminate between NK₂ tachykinin receptor subtypes

1990 • 174 citations

Actions of betahistine at histamine receptors in the brain

1985 • 157 citations

Behavioral and radioligand binding evidence for irreversible dopamine receptor blockade by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline

1983 • 135 citations

Atropine‐resistant longitudinal muscle spasms due to excitation of non‐cholinergic neurones in Auerbach's plexus

1968 • 128 citations

Inhibition of guinea pig ileum contractions mediated by a class of histamine receptor resembling the H3 subtype.

1987 • 117 citations

Histamine H₃‐receptors inhibit cholinergic neurotransmission in guinea‐pig airways

1989 • 110 citations

Effect of 5‐HT₃ receptor antagonists on responses to selective activation of mesolimbic dopaminergic pathways in the rat

1990 • 109 citations

Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?

1990 • 92 citations

N-carboxylic acid esters of 1,2- and 1,4-dihydroquinolines. New class of irreversible inactivators of the catechol amine .alpha.-receptors and potent central nervous system depressants

1968 • 91 citations

The mechanism of irreversible adrenergic blockade by N-carbethoxydihydroquinolines—model studies with typical serine hydrolases

1969 • 84 citations

Histamine H3-receptors modulate nonadrenergic noncholinergic neural bronchoconstriction in guinea-pig in vivo

1989 • 81 citations

Characterization of histamine H₃‐receptors in guinea‐pig ileum with H₃‐selective ligands

1990 • 75 citations

Effects of histamine H₁‐, H₂‐ and H₃‐receptor selective drugs on the mechanical activity of guinea‐pig small and large intestine

1991 • 71 citations

Inhibition of electrically evoked contractions of guinea-pig ileum preparations mediated by the histamine H3 receptor

1990 • 48 citations

Analysis of dose-response curves and calculation of agonist dissociation constants using a weighted nonlinear curve fitting program

1983 • 46 citations

Biexponential Kinetics of (R)‐α‐[³H]Methylhistamine Binding to the Rat Brain H₃ Histamine Receptor

1990 • 38 citations

Cholera and pertussis toxins amplify prostacyclin synthesis in aortic smooth muscle cells

1989 • 37 citations

Evidence for the existence of another type of histamine H2-receptor in guinea-pig ileum

1979 • 31 citations

Errors in agonist affinity estimation: do they and should they occur in isolated tissue experiments?

1990 • 30 citations

In Vitro and In Vivo Irreversible Blockade of Cortical S₂ Serotonin Receptors by N‐Ethoxycarbonyl‐2‐Ethoxy‐1,2‐Dihydroquinoline: A Technique for Investigating S₂ Serotonin Receptor Recovery

1986 • 30 citations

Receptors mediating the contractile response to neurokinin agonists in the guinea-pig trachea

1988 • 26 citations

Analysis of agonist action using the operational model

1988 • 25 citations

Characterisation of the Binding of the Histamine H3 Receptor Agonist [3H](R)-Alpha Methyl Histamine to Homogenates of Rat and Guinea-Pig Cortex

1991 • 25 citations

An inhibitory action of histamine on the guinea‐pig ileum

1970 • 23 citations

Mechanism of cholinergic antagonism by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ)

1970 • 20 citations

Antagonism by burimamide of inhibitions induced by histamine in plexus-containing longitudinal muscle preparations from guinea-pig ileum.

1973 • 19 citations