Carboxy terminus of vasopressin required for activity but not binding

pA, A NEW SCALE FOR THE MEASUREMENT OF DRUG ANTAGONISM

1947 • 759 citations

[1-(.beta.-mercapto-.beta.,.beta.-cyclopentamethylenepropionic acid),2-(O-methyl)tyrosine]arginine-vasopressin and [1-(.beta.-mercapto-.beta.,.beta.-cyclopentamethylenepropionic acid)]arginine-vasopressin, two highly potent antagonists of the vasopressor response to arginine-vasopressin

1980 • 449 citations

Frontiers in neuroendocrinology

1979 • 361 citations

ENZYMATIC CLEAVAGE OF GLYCINAMIDE FROM VASOPRESSIN AND A PROPOSED STRUCTURE FOR THIS PRESSOR-ANTIDIURETIC HORMONE OF THE POSTERIOR PITUITARY

1953 • 269 citations

A Major Metabolite of Arginine Vasopressin in the Brain Is a Highly Potent Neuropeptide

1983 • 261 citations

DIFFERENCES IN THE ANTIDIURETIC RESPONSES OF RATS TO THE INTRAVENOUS ADMINISTRATIONOF LYSINE AND ARGININE VASOPRESSINS¹

1958 • 120 citations

Vasopressin Analogs That Antagonize Antidiuretic Responses by Rats to the Antidiuretic Hormone

1981 • 114 citations

Neurohypophysial peptides design of tissue-specific agonists and antagonists

1981 • 99 citations

Design and uses of selective agonistic and antagonistic analogs of the neuropeptides oxytocin and vasopressin

1984 • 97 citations

Design of more potent antagonists of the antidiuretic responses to arginine-vasopressin

1982 • 78 citations

Synthetic antagonists of in vivo antidiuretic and vasopressor responses to arginine-vasopressin

1981 • 76 citations

Hormonally Active Arginine-Vasopressin Suppresses Endotoxin-Induced Fever in Rats: Lack of Effect of Oxytocin and a Behaviorally Active Vasopressin Fragment

1983 • 64 citations

Design of more potent and selective antagonists of the antidiuretic responses to arginine-vasopressin devoid of antidiuretic agonism

1982 • 49 citations

[8-Arginine]-Vasopressinoic Acid: An Inhibitor of Rabbit Kidney Adenyl Cyclase

1970 • 42 citations

[1-.beta.-Mercapto-.beta.,.beta.-diethylpropionic acid]-8-lysine-vasopressin, a potent inhibitor of 8-lysine-vasopressin and of oxytocin

1974 • 38 citations

Potent antagonists of the antidiuretic responses to arginine-vasopressin based on modifications of [1-(.beta.-mercapto-.beta.,.beta.-cyclopentamethylenepropionic acid),2-D-phenylalanine,4-valine]arginine-vasopressin at position four

1983 • 36 citations