Biochemical characterization of the interaction of three pyridazinyl-GABA derivatives with the GABAA receptor site

Benzodiazepine receptors in rat brain

1977 • 1,459 citations

GABAergic modulation of benzodiazepine binding site sensitivity

1978 • 726 citations

Bicuculline, an antagonist of GABA and synaptic inhibition in the spinal cord of the cat

1971 • 685 citations

Properties of γ-aminobutyric acid (GABA) receptor binding in rat brain synaptic membrane fractions

1975 • 637 citations

Binding characteristics of a radiolabeled agonist and antagonist at central nervous system alpha noradrenergic receptors.

1977 • 544 citations

Antiepileptic drugs : mechanisms of action

1980 • 508 citations

Influences ions, enzymes, and detergents on gamma-aminobutyric acid-receptor binding in synaptic membranes of rat brain.

1977 • 384 citations

Characteristics of GABA_B receptor binding sites on rat whole brain synaptic membranes

1983 • 377 citations

Characteristics of central 5-HT receptors and their adaptive changes following intracerebral 5,7-dihydroxytryptamine administration in the rat.

1978 • 336 citations

Characteristics of GABA_B receptor binding sites on rat whole brain synaptic membranes

1997 • 294 citations

Gaba agonists and antagonists

1979 • 222 citations

Stimulation of benzodiazepine receptor binding by gamma-aminobutyric acid.

1979 • 220 citations

THE EFFECT OF 4‐AMINO HEX‐5‐YNOIC ACID (γ‐ACETYLENIC GABA, γ‐ETHYNYL GABA) A CATALYTIC INHIBITOR OF GABA TRANSAMINASE, ON BRAIN GABA METABOLISM IN VIVO

1977 • 216 citations

3H-spiroperidol labels serotonin receptors in rat cerebral cortex and hippocampus

1978 • 206 citations

Distribution of glutamete decar☐ylase in discrete brain nuclei

1976 • 200 citations

Binding Characteristics and Interactions of Depressant Drugs with [³⁵S]t-Butylbicyclophosphorothionate, a Ligand that Binds to the Picrotoxinin Site

1984 • 156 citations

gamma-Aminobutyric acid receptor binding in mammalian brain. Heterogeneity of binding sites.

1981 • 150 citations

The Glycine Synaptic Receptor: Evidence That Strychnine Binding Is Associated with the Ionic Conductance Mechanism

1974 • 136 citations

Securinine alkaloids: A new class of GABA receptor antagonist

1985 • 121 citations

Characterization of specific, high-affinity binding sites for l-[3H]glutamic acid in rat brain membranes

1980 • 107 citations

Convulsant drugs: mechanisms of action.

1980 • 99 citations

Chemical instability of the GABA antagonist bicuculline under physiological conditions

1975 • 89 citations

A steroid derivative, R 5135, antagonizes the GABA/benzodiazepine receptor interaction

1981 • 88 citations

GABA binding in mammalian brain: Inhibition by endogenous GABA

1980 • 81 citations

Na+-independent binding of GABA to the triton X-100 treated synaptic membranes from cerebellum of rat brain

1977 • 78 citations

An arylaminopyridazine derivative of gamma-aminobutyric acid (GABA) is a selective and competitive antagonist at the GABAA receptor site.

1985 • 78 citations

Pitrazepin, a novel GABAA antagonist

1984 • 63 citations

Antagonism between bicuculline, strychnine, and picrotoxin and depressant amino-acids in the rat nervous system

1972 • 62 citations

N-Ethylmaleimide-induced alteration in the interaction of agonists with muscarinic cholinergic receptors of rat brain.

1983 • 53 citations

Interactions between three pyridazinyl-GABA derivatives and central GABA and glycine receptors in the rat, an in vivo microiontophoretic study

1986 • 39 citations

Developmental studies of the uptake of choline, gaba and dopamine by crude synaptosomal preparations after in vivo or in vitro lead treatment

1980 • 35 citations

Stereospecific interaction of bicuculline with specific [3H]strychnine binding to rat spinal cord synaptosomal membranes

1980 • 33 citations

Binding of [³H] γ‐Aminobutyric Acid and [³H]Muscimol in Purified Rat Brain Synaptic Plasma Membranes and the Effects of Bicuculline

1982 • 31 citations

Effect of picrotoxin on benzodiazepine receptors and GABA receptors with reference to the effect of Cl− ion

1981 • 30 citations

GABA agonists and potential antagonists related to muscimol

1979 • 27 citations

Diazotization and Thiocyanate Differentiate Agonists from Antagonists for the High‐ and Low‐Affinity Receptors of γ‐Aminobutyric Acid

1984 • 26 citations