General synthetic access to α-allenyl amines and α-allenyl-α-aminoacids as potential enzyme activated irreversible inhibitors of PLP dependent enzymes

Catalytic irreversible inhibition of mammalian ornithine decarboxylase (E.C.4.1.1.17) by substrate and product analogs

1978 • 998 citations

Selective inhibitors of biosynthesis of aminergic neurotransmitters

1978 • 424 citations

4‐Amino‐hex‐5‐enoic Acid, a Selective Catalytic Inhibitor of 4‐Aminobutyric‐Acid Aminotransferase in Mammalian Brain

1977 • 375 citations

Efficient homologation of acetylenes to allenes

1979 • 164 citations

Acetylenic enzyme inactivators. Inactivation of .gamma.-cystathionase, in vitro and in vivo by propargylglycine

1973 • 139 citations

Regiospecific 1,4 addition of a propargylic anion. A general synthon for 2-substituted propargylamines as potential catalytic irreversible enzyme inhibitors.

1975 • 73 citations

Hetero Cope Rearrangements in the Cyclization of Allyl and Propargyl Esters of N‐Acyl Amino Acids to Oxazolin‐5‐ones

1975 • 66 citations

Mechanism of inactivation of γ-cystathionase by β,β,β-trifluoroalanine

1977 • 45 citations

Trimethylsilylacetylene-N-carboethoxy glycinate dianion - a general synthon for α-acetylenic α-amino acids.

1978 • 41 citations

Synthesis of β,γ-unsaturated amino acids as potential catalytic irreversible enzyme inhibitors

1977 • 38 citations

Synthese d'amino-alcools alleniques.

1982 • 23 citations

Syntheses of α-ethynyl-3, 4-dihydroxyphenylalanine and α-vinyl-3, 4-dihydroxyphenylalanine

1977 • 16 citations

Une methode generale de synthese d'allenes fonctionnalises en α

1978 • 16 citations

Stereospecific irreversible inhibition of mammalian (S)-ornithine decarboxylase by (R)-(–)-hex-5-yne-1,4-diamine

1982 • 16 citations