Comparison of the In-vitro Receptor Selectivity of Substituted Benzamide Drugs for Brain Neurotransmitter Receptors

Specific in vitro and in vivo binding of 3H-raclopride a potent substituted benzamide drug with high affinity for dopamine D-2 receptors in the rat brain

1985 • 503 citations

Remoxipride, a new potential antipsychotic compound with selective anti-dopaminergic actions in the rat brain

1984 • 213 citations

Dopamine Receptor Parameters Detected by [³H]Spiperone Depend on Tissue Concentration: Analysis and Examples

1984 • 173 citations

Substituted benzamide drugs as selective neuroleptic agents.

1981 • 122 citations

Dopamine D2 receptors selectively labeled by a benzamide neuroleptic: [3H]-YM-09151-2

1985 • 108 citations

Selective binding of YM-09151-2, a new potent neuroleptic, to D2-dopaminergic receptors.

1983 • 103 citations

Effects of Remoxipride and some Related New Substituted Salicylamides on Rat Brain Receptors

1986 • 101 citations

[]-N-: The radioligand of choice for pett studies of the dopamine receptor in human brain

1985 • 97 citations

DOPAMINE RECEPTOR BLOCKING ACTIVITY OF SULPIRIDE IN THE CENTRAL NERVOUS SYSTEM

1977 • 92 citations

Specific binding of [3H]sulpiride to rat striatal preparations

1979 • 87 citations

In vivo quantitative imaging of dopamine receptors in human brain using positron emission tomography and [76Br]bromospiperone

1985 • 77 citations

Comparison of dopamine receptor sites labeled by [3H]-S-sulpiride and [3H]-spiperone in striatum.

1983 • 70 citations

Neuroleptic properties of cis-N-(1-benzyl-2-methylpyrrolidin-3-yl)-5-chloro-2-methoxy-4-methylaminobenzamide (YM-09151-2) with selective antidopaminergic activity

1981 • 65 citations

3-N-(2-[18F]-fluoroethyl)-spiperone: A novel ligand for cerebral dopamine receptor studies with pet

1987 • 62 citations

Binding of [3H]sulpiride to purified rat striatal synaptic membranes

1981 • 47 citations

Assessment of dopamine receptor densities in the human brain with carbon-11-labeled N-methylspiperone

1984 • 42 citations

Review on neuroleptic receptors: specificity and multiplicity of in vitro binding related to pharmacological activity

1981 • 24 citations

SELECTIVE BINDING OF YM-09151-2, A NEW POTENT NEUROLEPTIC, TO D2-DOPAMINERGIC RECEPTORS

1983 • 19 citations

Pharmacological characterization of binding sites identified in rat brain following in vivo administration of [³H]‐spiperone.

1987 • 12 citations

Definition of the In-vivo Accumulation of [3H]spiperone in Brain using Haloperidol and Sulpiride to Determine Functional Dopamine Receptor Occupation

1988 • 5 citations

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