[3H]Harman Binding Experiments. I: A Reversible and Selective Radioligand for Monoamine Oxidase Subtype A in the CNS of the Rat

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1973 • 12,522 citations

Some observations upon a new inhibitor of monoamine oxidase in brain tissue

1968 • 1,589 citations

A rapid microfluorimetric determination of monoamine oxidase

1965 • 406 citations

Isatin: Identity with the Purified Endogenous Monoamine Oxidase Inhibitor Tribulin

1988 • 202 citations

The Synaptosome

1969 • 197 citations

Ethnopharmacologic Search for Psychoactive Drugs.

1980 • 180 citations

Monoamine oxidase inhibition in brain and liver produced by β-carbolines: structure-activity relationships and substrate specificity

1977 • 180 citations

Differential Changes in Monoamine Oxidase A and B Activity in the Aging Rat Brain

1980 • 173 citations

Interactions of monoamine oxidase with substrates and inhibitors

1989 • 141 citations

Criteria for receptor sites in binding studies

1984 • 128 citations

Benzodiazepine antagonism by harmane and other β-carbolines in vitro and in vivo

1981 • 124 citations

1-Methyl-?-carboline (Harmane), a potent endogenous inhibitor of benzodiazepine receptor binding

1980 • 119 citations

The nature of the inhibition of rat liver monoamine oxidase types A and B by the acetylenic inhibitors clorgyline, l-deprenyl and pargyline

1982 • 117 citations

Additional evidence for the existence of several forms of mitochondrial monoamine oxidase in the mouse

1968 • 97 citations

Stereoselectivity and isoenzyme selectivity of monoamine oxidase inhibitors

1985 • 92 citations

[³H]Propyl ?-Carboline-3-Carboxylate Binds Specifically to Brain Benzodiazepine Receptors

1981 • 89 citations

[³H]HARMALINE AS A SPECIFIC LIGAND OF MAO A—I. PROPERTIES OF THE ACTIVE SITE OF MAO A FROM RAT AND BOVINE BRAINS

1979 • 76 citations

The monoamine oxidase inhibiting properties of CGP 11305 A

1983 • 71 citations

Tetrahydroisoquinolines and β-carbolines: putative natural substances in plants and mammals

1985 • 69 citations

Identification of harman in the rat arcuate nucleus

1980 • 61 citations

Kinetic studies and effects in vivo of a new monoamine oxidase inhibitor, N[2(ochlorophenoxy)-ethyl]-cyclopropylamine

1968 • 61 citations

?-Carbolines as selective monoamine oxidase inhibitors:In vivo implications

1982 • 59 citations

TETRAHYDRO‐β‐CARBOLINES: SPECIFIC INHIBITORS OF TYPE A MONOAMINE OXIDASE IN RAT BRAIN¹

1977 • 58 citations

Binding of [³H]DMCM, a Convulsive Benzodiazepine Ligand, to Rat Brain Membranes: Preliminary Studies

1983 • 52 citations

Synthesis Experiments in the Group of Hypotensive Alkaloids--XXI. Chemistry of 1,2,3,4-Tetra-hydronorharmane-1-carboxylic Acid and Derivatives

1961 • 51 citations

5‐HYDROXYTRYPTAMINE CATABOLISM IN THE RAT BRAIN DURING ONTOGENESIS

1977 • 45 citations

Properties of agonist binding at the?-adrenoceptor of the rat reticulocyte

1982 • 44 citations

High affinity (3H)tryptamine binding sites in various organs of the rat

1984 • 41 citations

Harman in rat brain, lung and human CSF: Effect of alcohol consumption

1988 • 39 citations

Demonstration of a distinct class of high-affinity binding sites for [3H]norharman ([3H]β-carboline) in the rat brain

1988 • 35 citations

[³H]Harman Binding Experiments. II: Regional and Subcellular Distribution of Specific [³H]Harman Binding and Monoamine Oxidase Subtypes A and B Activity in Marmoset and Rat

1991 • 34 citations

Characteristics of the Inhibition of Rat Brain Monoamine Oxidase In Vitro by MD780515

1981 • 32 citations

Properties of [3H] ß-carboline-3-carboxylate ethyl ester binding to the benzodiazepine receptor

1981 • 31 citations

Design and early clinical evaluation of selective inhibitors of monoamine oxidase

1988 • 31 citations

[³H]HARMALINE AS A SPECIFIC LIGAND OF MAO A–II. MEASUREMENT OF THE TURNOVER RATES OF MAO A DURING ONTOGENESIS IN THE RAT BRAIN

1979 • 30 citations

Monoamine oxidase A from human placenta and monoamine oxidase B from bovine liver both have one FAD per subunit

1989 • 30 citations

On the inhibition by harmine of oxidative deamination of biogenic monoamines

1967 • 26 citations

Quantitative autoradiography of [3H]norharman [( 3H]beta-carboline) binding sites in the rat brain.

1990 • 22 citations

Specific 3H-DMCM binding to a non-benzodiazepine binding site after silver ion treatment of rat brain membranes

1984 • 4 citations

Non-benzodiazepine, Ag-dependent, brain-specific binding sites for [3H] β-carboline-3-carboxylic acid ethyl ester

1989 • 1 citations

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