Comparative binding of μ and δ selective ligands in whole brain and pons/medulla homogenates from rat: Affinity profiles of fentanyl derivatives

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1973 • 12,522 citations

REGIONAL STUDIES OF CATECHOLAMINES IN THE RAT BRAIN‐I

1966 • 5,429 citations

Quantitative analysis of drug-receptor interactions: I. Determination of kinetic and equilibrium properties

1981 • 557 citations

SPECTRUM OF THE μ‐, δ‐ AND κ‐BINDING SITES IN HOMOGENATES OF RAT BRAIN

1982 • 278 citations

Separation of opioid analgesia from respiratory depression: evidence for different receptor mechanisms.

1985 • 271 citations

Opioids and breathing

1985 • 171 citations

The use of [³H]‐[<scp>d</scp>‐Pen²,<scp>d</scp>‐Pen⁵]enkephalin as a highly selective ligand for the δ‐binding site

1985 • 99 citations

Species differences in the concentrations and distributions of opioid binding sites

1985 • 99 citations

Potent, New Analgesics, Tailor‐Made for Different Purposes

1982 • 78 citations

Multiple mu opiate receptors: Biochemical and pharmacological evidence for multiplicity

1986 • 77 citations

[D-Pen2,D-Pen5]enkephalin (DPDPE): a δ-selective enkephalin with low affinity for μ1 opiate binding sites

1986 • 53 citations

A comparative study in rats of the respiratory depression and analgesia induced by μ- and δ-opioid agonists

1984 • 30 citations

Binding properties of 3H-lofentanil at the opiate receptor.

1982 • 13 citations

Determination of proenkephalin products in brain tissue by high-performance liquid chromatography and a modified bioassay procedure

1985 • 9 citations

Failure to demonstrate mu-isoreceptors

1984 • 6 citations

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