5β-Pregnan-3β-ol-20-one, a specific antagonist at the neurosteroid site of the GABAA receptor-complex

Structure-activity relationships for steroid interaction with the gamma-aminobutyric acidA receptor complex.

1987 • 601 citations

The neurosteroid dehydroepiandrosterone sulfate is an allosteric antagonist of the GABAA receptor

1990 • 433 citations

Pregnenolone-sulfate: an endogenous antagonist of the γ-aminobutyric acid receptor complex in brain?

1987 • 329 citations

Characterization of steroid interactions with gamma-aminobutyric acid receptor-gated chloride ion channels: evidence for multiple steroid recognition sites.

1990 • 328 citations

Modulation of the GABA_A receptor by depressant barbiturates and pregnane steroids

1988 • 296 citations

Steroid anesthetics and naturally occurring analogs modulate the gamma-aminobutyric acid receptor complex at a site distinct from barbiturates.

1989 • 266 citations

GABAA receptor subtypes immunopurified from rat brain with α subunit-specific antibodies have unique pharmacological properties

1991 • 195 citations

Physiological aspects of steroids with anaesthetic properties.

1976 • 78 citations

Action of Some Steroids on the Central Nervous System of the Mouse. II. Pharmacology

1965 • 78 citations

Antagonist-type interaction of glucocorticoids with the GABA receptor-coupled chloride channel

1987 • 75 citations

Neuroendocrine Metabolism of Progesterone and Related Progestins

2007 • 72 citations

Modulation of the GABA_A receptor complex by steroids in slices of rat cuneate nucleus

1989 • 71 citations

Steroids and neuronal activity

1991 • 26 citations

The stimulatory effects of secobarbital and pregnanolone on the GABAA receptor can be blocked selectively

1988 • 25 citations