GABAB receptor antagonists: from synthesis to therapeutic applications
Data up to Jan 2025
Total Citations Per Year
Abstract
References (16)
A physiological role for GABAB receptors in the central nervous system
1988 • 643 citations
The Role of GABA B Receptor Activation in Absence Seizures of Lethargic ( lh / lh ) Mice
1992 • 355 citations
Phaclofen: a peripheral and central baclofen antagonist
1987 • 349 citations
CGP 35348: a centrally active blocker of GABAB receptors
1990 • 303 citations
2-Hydroxy-saclofen: an improved antagonist at central and peripheral GABAB receptors
1988 • 202 citations
Upregulation of gamma-aminobutyric acid (GABA) B binding sites in rat frontal cortex: a common action of repeated administration of different classes of antidepressants and electroshock.
1985 • 197 citations
GABAB receptors in mammalian function
1991 • 146 citations
CGP 36742: The first orally active GABAB blocker improves the cognitive performance of mice, rats, and rhesus monkeys
1993 • 119 citations
The actions of orally active GABAB receptor antagonists on GABAergic transmission in vivo and in vitro
1993 • 92 citations
CGP 35348, a new GABAB antagonist, prevents antinociception and muscle‐relaxant effect induced by baclofen
1991 • 73 citations
Functional evidence for multiple gamma-aminobutyric acidB receptor subtypes in the rat cerebral cortex.
1992 • 72 citations
Repeated administration of desipramine and a GABAB receptor antagonist, CGP 36742, discretely up‐regulates GABAB receptor binding sites in rat frontal cortex
1993 • 64 citations
Are increases in GABAB receptors consistent findings following chronic antidepressant administration?
1987 • 53 citations
Phaclofen: a GABAB blocker reduces long-duration inhibition in the neocortex
1988 • 42 citations
Inhibition of baolofen-induced hypothermia in mice by the novel GABAB antagonist CGP 35348
1991 • 25 citations
Increased acetylcholine and quisqualate responsiveness after blockade of GABAB receptors
1992 • 23 citations