Contractile 5‐HT1B receptors in human cerebral arteries: pharmacological characterization and localization with immunocytochemistry
Data up to Jan 2025
Total Citations Per Year
Abstract
References (39)
International Union of Pharmacology classification of receptors for 5-hydroxytryptamine (Serotonin).
1994 • 2,935 citations
Brain stem activation in spontaneous human migraine attacks
1995 • 1,366 citations
Hypothalamic activation in cluster headache attacks
1998 • 1,098 citations
pA2 and receptor differentiation: A statistical analysis of competitive antagonism
1979 • 408 citations
Mechanical properties of rat cerebral arteries as studied by a sensitive device for recording of mechanical activity in isolated small blood vessels*
1983 • 402 citations
Migraine pain associated with middle cerebral artery dilatation: reversal by sumatriptan
1991 • 376 citations
GR43175, a selective agonist for the 5‐HT1‐like receptor in dog isolated saphenous vein
1988 • 305 citations
Human serotonin 1D receptor is encoded by a subfamily of two distinct genes: 5-HT1D alpha and 5-HT1D beta.
1992 • 293 citations
A single amino-acid difference confers major pharmacological variation between human and rodent 5-HT1B receptors
1992 • 279 citations
Mode of action of the anti-migraine drug sumatriptan
1991 • 249 citations
A subfamily of 5-HT1D receptor genes
1992 • 230 citations
Differential Distribution of 5Ht1D-and 5HT1B-Immunoreactivity within the Human Trigemino-Cerebrovascular System: Implications for the Discovery of New Antimigraine Drugs
1997 • 225 citations
Primary structure and functional characterization of a human 5-HT1D-type serotonin receptor.
1991 • 225 citations
Characterization of the human 5-hydroxytryptamine1B receptor.
1992 • 172 citations
Differential expression of sumatriptan-sensitive 5-hydroxytryptamine receptors in human trigeminal ganglia and cerebral blood vessels.
1996 • 171 citations
5‐HT1‐like receptors mediate 5‐hydroxytryptamine‐induced contraction of human isolated basilar artery
1989 • 169 citations
Variable participation of 5-HT1-like receptors and 5-HT2 receptors in serotonin-induced contraction of human isolated coronary arteries. 5-HT1-like receptors resemble cloned 5-HT1D beta receptors.
1994 • 167 citations
Sumatriptan (GR 43175) interacts selectively with 5-HT1B and 5-HT1D binding sites
1989 • 160 citations
5-HT1F receptor agonists inhibit neurogenic dural inflammation in guinea pigs
1997 • 158 citations
Pharmacological analysis of 5-hydroxytryptamine receptors in isolated intracranial and extracranial vessels of cat and man.
1978 • 156 citations
Evidence for 5-HT1B/1D Receptors Mediating the Antimigraine Effect of Sumatriptan and Dihydroergotamine
1991 • 153 citations
Expression of mRNA for the serotonin 5-hydroxytryptamine1D beta receptor subtype in human and bovine cerebral arteries.
1993 • 136 citations
Selective 5-HT1D alpha serotonin receptor gene expression in trigeminal ganglia: implications for antimigraine drug development.
1994 • 126 citations
Naratriptan
1997 • 123 citations
Receptor specificity and trigemino‐vascular inhibitory actions of a novel 5‐HT1B/1D receptor partial agonist, 311C90 (zolmitriptan)
1997 • 99 citations
Vasoconstriction in human isolated middle meningeal arteries: determining the contribution of 5‐HT1B‐ and 5‐HT1F‐receptor activation
1999 • 97 citations
A human serotonin 1D receptor variant (5HT1D beta) encoded by an intronless gene on chromosome 6.
1992 • 95 citations
The selective closure of feline carotid arteriovenous anastomoses (AVAs) by GR43175
1989 • 83 citations
Comparison of the vasoconstrictor effects of rizatriptan and sumatriptan in human isolated cranial arteries: immunohistological demonstration of the involvement of 5‐HT1B‐receptors
1998 • 83 citations
5‐HT1 receptors in migraine pathophysiology and treatment
1995 • 79 citations
Contractile 5‐HT1 receptors in human isolated pial arterioles: correlation with 5‐HT1D binding sites
1991 • 78 citations
Molecular cloning of a human serotonin receptor (S12) with a pharmacological profile resembling that of the 5-HT1D subtype.
1992 • 75 citations
Sumatriptan is a Potent Vasoconstrictor of Human Dural Arteries Via a 5-HT1-Like Receptor
1992 • 69 citations
5‐HT1B receptor‐mediated contractions in human temporal artery: evidence from selective antagonists and 5‐HT receptor mRNA expression
1998 • 68 citations
Migraine Pharmacology and Genetics
1997 • 54 citations
5‐Hydroxytryptamine receptor characterizations of human cerebral, middle meningeal and temporal arteries: regional differences
1993 • 49 citations
Endothelial expression of the 5-hydroxytryptamine1B antimigraine drug receptor in rat and human brain microvessels
1998 • 39 citations
Participation of 5‐HT1‐like and 5‐HT2A receptors in the contraction of human temporal artery by 5‐hydroxytryptamine and related drugs
1996 • 27 citations
Assessment of Peripheral Vascular Effects of Antimigraine Drugs in Humans
1995 • 20 citations