Solid-Phase Synthesis of a 6-Phenylquinolin-2(1H)-one Library Directed toward Nuclear Hormone Receptors

Nuclear Hormone Receptors and Gene Expression

2001 • 1,538 citations

Nuclear-Receptor Ligands and Ligand-Binding Domains

1999 • 314 citations

Androgen Receptor Antagonists (Antiandrogens) Structure-Activity Relationships

2000 • 225 citations

Pharmacological Options in the Treatment of Benign Prostatic Hyperplasia

1997 • 169 citations

Synthesis and Biological Activity of a Novel Series of Nonsteroidal, Peripherally Selective Androgen Receptor Antagonists Derived from 1,2-Dihydropyridono[5,6-g]quinolines

1998 • 140 citations

Discovery of a Potent, Orally Active, Nonsteroidal Androgen Receptor Agonist: 4-Ethyl-1,2,3,4-tetrahydro-6- (trifluoromethyl)-8-pyridono[5,6-g]- quinoline (LG121071)

1999 • 85 citations

6-Substituted 1H-quinolin-2-ones and 2-methoxy-quinolines: Synthesis and evaluation as inhibitors of steroid 5α reductases types 1 and 2

2000 • 51 citations

Synthesis, SAR and in vivo activity of novel thienopyridine sulfonamide pyrrolidinones as factor Xa inhibitors

1999 • 25 citations