Chemical modification and irreversible inhibition of striatal A2a adenosine receptors.

[41] Modification of histidyl residues in proteins by diethylpyrocarbonate

1977 • 813 citations

Cardiovascular purinoceptors

1990 • 666 citations

Selective Amplification And Cloning Of Four New Members Of The G Protein-coupled Receptor Family

1989 • 647 citations

[3H]CGS 21680, a selective A2 adenosine receptor agonist directly labels A2 receptors in rat brain.

1989 • 537 citations

The adenosine/neutrophil paradox resolved: human neutrophils possess both A1 and A2 receptors that promote chemotaxis and inhibit O2 generation, respectively.

1990 • 377 citations

RDC8 codes for an adenosine A2 receptor with physiological constitutive activity

1990 • 270 citations

Cloning and expression of an A1 adenosine receptor from rat brain.

1991 • 235 citations

Adenosine A₁ and A₂ receptors: Structure–function relationships

1992 • 126 citations

Distinct pathways of desensitization of A1- and A2-adenosine receptors in DDT1 MF-2 cells.

1991 • 126 citations

A2A adenosine receptors from rat striatum and rat pheochromocytoma PC12 cells: characterization with radioligand binding and by activation of adenylate cyclase.

1992 • 115 citations

Behavioral effects of A1- and A2-selective adenosine agonists and antagonists: evidence for synergism and antagonism.

1991 • 103 citations

Identification of the A2 adenosine receptor binding subunit by photoaffinity crosslinking.

1989 • 81 citations

Neuere Methoden der präparativen organischen Chemie

1941 • 80 citations

Separation of solubilized A2 adenosine receptors of human platelets from non-receptor [3H]NECA binding sites by gel filtration

1988 • 70 citations

The A2 adenosine receptor: guanine nucleotide modulation of agonist binding is enhanced by proteolysis.

1991 • 58 citations

Chemical modification of A1 adenosine receptors in rat brain membranes. Evidence for histidine in different domains of the ligand binding site.

1988 • 51 citations

Agonist derived molecular probes for A₂ adenosine receptors

1989 • 37 citations

Electrophilic derivatives of purines as irreversible inhibitors of A1 adenosine receptors

1989 • 35 citations

High affinity acylating antagonists for the A1 adenosine receptor: identification of binding subunit.

1988 • 31 citations

Kinetics and mechanism of the Bamberger cleavage of imidazole and of histidine derivatives by diethyl pyrocarbonate in aqueous solution

1980 • 24 citations

Evidence for the participation of histidine residues located in the 56 kDa C‐terminal polypeptide domain of ADP‐ribosyl transferase in its catalytic activity

1990 • 22 citations

Probing the adenosine receptor with adenosine and xanthine biotin conjugates

1985 • 22 citations

Chemical modification of adenosine A1 receptors

1990 • 19 citations

Trifunctional agents as a design strategy for tailoring ligand properties: irreversible inhibitors of A1 adenosine receptors

1991 • 15 citations

Inhibition of muscarinic cholinergic receptors by disulfide reducing agents and arsenicals

1991 • 14 citations

[3H]XAC (xanthine amine congener) is a radioligand for A2-adenosine receptors in rabbit striatum

1991 • 11 citations

Thermal Fragmentations. VI. The Preparation of Aryl N-Monoalkyldithiocarbamates and Their Behaviour Upon Heating.

1973 • 6 citations